SCHEMBL6140590

SCHEMBL6140590

COc1cccc(OC)c1C(=O)[AsH]C(Cc1ccc2nc(-c3c(Cl)cccc3Cl)ccc2c1)C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 11/20 0.56
ITGAV P06756 1/20 0.56
ITGA4 P13612 10/20 0.36
ITGB7 P26010 6/20 0.36
ABL1 P00519 1/20 0.35
FABP4 P15090 1/20 0.34
LDHA P00338 1/20 0.34
CCR2 P41597 1/20 0.34
CTSA P10619 1/20 0.33
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6140931 0.93 ITGB1 (0.54) ITGB1ITGAVITGA4ITGB7LDHA
SCHEMBL6142370 0.90 ITGB1 (0.66) ITGB1ITGAVITGA4ITGB7ABL1
SCHEMBL6141516 0.85 ITGB1 (0.51) ITGB1ITGAVITGA4ITGB7
SCHEMBL3317055 0.82 ITGB1 (0.81) ITGB1ITGAVITGA4ITGB7
SCHEMBL6141061 0.81 ITGB1 (0.55) ITGB1ITGAVITGA4ITGB7ABL1
SCHEMBL6141364 0.81 EIF4E (0.38) ITGB1ITGAV
SCHEMBL6146195 0.80 ITGB1 (0.54) ITGB1ITGAVITGA4ITGB7ABL1
SCHEMBL6141873 0.79 ITGB1 (0.53) ITGB1ITGAVITGA4ITGB7ABL1
SCHEMBL6151313 0.79 ITGB1 (0.52) ITGB1ITGAVITGA4ITGB7
SCHEMBL6142182 0.77 ITGB1 (0.47) ITGB1ITGAVITGA4ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2005-02-02 EP claimed
WO-2003093237-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2003-11-13 WO claimed