SCHEMBL6151313

SCHEMBL6151313

O=C([AsH]C(Cc1ccc2nc(-c3ccncc3)ccc2c1)C(=O)O)c1c(Cl)cccc1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 5/20 0.52
ITGAV P06756 2/20 0.52
KCNH2 Q12809 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
ITGA4 P13612 3/20 0.36
ITGB7 P26010 3/20 0.36
CYP2C9 P11712 2/20 0.36
NPC1 O15118 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
AR P10275 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
RAB9A P51151 1/20 0.36
MAPT P10636 1/20 0.35
BLM P54132 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
MAPK1 P28482 1/20 0.33
DOT1L Q8TEK3 1/20 0.33
MPL P40238 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6142370 0.88 ITGB1 (0.66) ITGB1ITGAVKCNH2HRH3ITGA4
SCHEMBL6140931 0.82 ITGB1 (0.54) ITGB1ITGAVITGA4ITGB7
SCHEMBL3313527 0.81 ITGB1 (0.79) ITGB1ITGAVITGA4ITGB7
SCHEMBL6140590 0.79 ITGB1 (0.56) ITGB1ITGAVITGA4ITGB7
SCHEMBL6140902 0.77 ITGB1 (0.44) ITGB1ITGAVITGA4ITGB7
SCHEMBL6141873 0.76 ITGB1 (0.53) ITGB1ITGAVKCNH2HRH3ITGA4
SCHEMBL6141516 0.74 ITGB1 (0.51) ITGB1ITGAVITGA4ITGB7RAB9A
SCHEMBL4409576 0.74 ITGB1 (0.85) ITGB1ITGAVITGA4ITGB7
SCHEMBL6142182 0.73 ITGB1 (0.47) ITGB1ITGAVKCNH2HRH3ITGA4
SCHEMBL6141061 0.72 ITGB1 (0.55) ITGB1ITGAVKCNH2HRH3ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2005-02-02 EP disclosed
WO-2003093237-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2003-11-13 WO disclosed