SCHEMBL6145239

SCHEMBL6145239

Cc1ccc(S(=O)(=O)N2[C@H](C(=O)[AsH]C(Cc3ccc4nc(-c5c(Cl)cccc5Cl)ccc4c3)C(=O)O)C[C@@H]3CCCC[C@@H]32)cc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 6/20 0.42
ITGAV P06756 1/20 0.42
ITGA4 P13612 5/20 0.37
MAPT P10636 1/20 0.34
ALDH1A1 P00352 3/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PLA2G1B P04054 1/20 0.34
PKM P14618 1/20 0.34
ATG4B Q9Y4P1 1/20 0.34
GAA P10253 1/20 0.34
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33
ITGB7 P26010 1/20 0.33
ABL1 P00519 1/20 0.32
FKBP1A P62942 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3317863 0.86 ITGB1 (0.53) ITGB1ITGAVITGA4ALDH1A1L3MBTL1
SCHEMBL4410500 0.86 ITGB1 (0.53) ITGB1ITGAVITGA4ALDH1A1L3MBTL1
SCHEMBL4625418 0.83 ITGB1 (0.44) ITGB1ITGAVITGA4MAPTALDH1A1
SCHEMBL3314360 0.79 ITGB1 (0.48) ITGB1ITGAVITGA4ALDH1A1L3MBTL1
SCHEMBL6142066 0.79 ITGB1 (0.45) ITGB1ITGAVITGA4MAPTALDH1A1
SCHEMBL3320849 0.75 ITGB1 (0.56) ITGB1ITGAVITGA4ALDH1A1L3MBTL1
SCHEMBL3318694 0.74 ITGB1 (0.45) ITGB1ITGAVITGA4ALDH1A1ITGB7
SCHEMBL4625253 0.74 ITGB1 (0.43) ITGB1ITGAVITGA4ALDH1A1ITGB7
SCHEMBL3313128 0.74 ITGB1 (0.43) ITGB1ITGAVITGA4ALDH1A1ITGB7
SCHEMBL6140359 0.72 ITGB1 (0.55) ITGB1ITGAVITGA4MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2005-02-02 EP claimed
WO-2003093237-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2003-11-13 WO claimed
EP-1501801-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2005-02-02 EP disclosed
WO-2003093237-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2003-11-13 WO disclosed