SCHEMBL6149013

SCHEMBL6149013

CCOC(=O)N1CCN(C(=O)OCCC2CCN(C(=O)NC[C@H](NC(=O)[C@H]3CCCN3S(=O)(=O)c3cc(Cl)cc(Cl)c3)C(=O)OC)CC2)CC1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 17/20 0.46
ITGA4 P13612 17/20 0.46
ITGA2 P17301 1/20 0.42
ITGB7 P26010 1/20 0.41
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
MMP1 P03956 1/20 0.38
MMP3 P08254 1/20 0.38
MMP7 P09237 1/20 0.38
MMP9 P14780 1/20 0.38
MMP13 P45452 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6149008 1.00 ITGB1 (0.46) ITGB1ITGA4ITGA2ITGB7HCRTR1
SCHEMBL6152677 0.94 ITGB1 (0.45) ITGB1ITGA4ITGA2ITGB7HCRTR1
SCHEMBL6401299 0.94 ITGA4 (0.49) ITGB1ITGA4ITGA2ITGB7MEN1
SCHEMBL6401304 0.94 ITGA4 (0.49) ITGB1ITGA4ITGA2ITGB7MEN1
SCHEMBL6149763 0.90 ITGB1 (0.43) ITGB1ITGA4ITGA2ITGB7HCRTR1
SCHEMBL6156097 0.90 ITGA4 (0.42) ITGB1ITGA4ITGA2ITGB7HCRTR1
SCHEMBL6152300 0.89 ITGB1 (0.48) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6152295 0.89 ITGB1 (0.48) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6149667 0.89 ITGB1 (0.48) ITGB1ITGA4ITGA2ITGB7
SCHEMBL6149675 0.89 ITGB1 (0.48) ITGB1ITGA4ITGA2ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1495044-A1 HETEROCYCLIC AMIDES WITH ALPHA-4 INTEGRIN ANTAGONIST ACTIVITY J. Uriach y Compania S.A. (ES) 2005-01-12 EP disclosed
WO-2003084984-A1 HETEROCYCLIC AMIDES WITH ALPHA-4 INTEGRIN ANTAGONIST ACTIVITY J. URIACH Y COMPANIA S.A. (ES) 2003-10-16 WO disclosed