SCHEMBL6152677

SCHEMBL6152677

COC(=O)[C@H](CNC(=O)N1CCC(CCOC(=O)N2CCC(C)CC2)CC1)NC(=O)C1CCCN1S(=O)(=O)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 19/20 0.45
ITGA4 P13612 19/20 0.45
ITGB7 P26010 2/20 0.41
ITGA2 P17301 1/20 0.40
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6149008 0.94 ITGB1 (0.46) ITGB1ITGA4ITGB7ITGA2HCRTR1
SCHEMBL6402881 0.94 ITGB1 (0.49) ITGB1ITGA4ITGB7ITGA2
SCHEMBL6404278 0.94 ITGB1 (0.49) ITGB1ITGA4ITGB7ITGA2
SCHEMBL6447885 0.94 ITGB1 (0.49) ITGB1ITGA4ITGB7ITGA2
SCHEMBL6149013 0.94 ITGB1 (0.46) ITGB1ITGA4ITGB7ITGA2HCRTR1
SCHEMBL6149763 0.92 ITGB1 (0.43) ITGB1ITGA4ITGB7ITGA2HCRTR1
SCHEMBL6156097 0.88 ITGA4 (0.42) ITGB1ITGA4ITGB7ITGA2HCRTR1
SCHEMBL6401304 0.88 ITGA4 (0.49) ITGB1ITGA4ITGB7ITGA2
SCHEMBL6401299 0.88 ITGA4 (0.49) ITGB1ITGA4ITGB7ITGA2
SCHEMBL6152295 0.88 ITGB1 (0.48) ITGB1ITGA4ITGB7ITGA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1495044-A1 HETEROCYCLIC AMIDES WITH ALPHA-4 INTEGRIN ANTAGONIST ACTIVITY J. Uriach y Compania S.A. (ES) 2005-01-12 EP disclosed
WO-2003084984-A1 HETEROCYCLIC AMIDES WITH ALPHA-4 INTEGRIN ANTAGONIST ACTIVITY J. URIACH Y COMPANIA S.A. (ES) 2003-10-16 WO disclosed