SCHEMBL6151165

SCHEMBL6151165

CCCC(NC(=O)[C@H]1CCCN1S(=O)(=O)c1ccc(C)cc1)C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 2/20 0.58
ITGB1 P05556 3/20 0.58
ITGA2 P17301 1/20 0.58
GAA P10253 1/20 0.57
HPGD P15428 1/20 0.57
FKBP1A P62942 1/20 0.56
L3MBTL1 Q9Y468 3/20 0.54
MAPK1 P28482 2/20 0.54
TSHR P16473 2/20 0.53
POLB P06746 1/20 0.53
ITGA5 P08648 2/20 0.52
MMP2 P08253 1/20 0.52
MMP9 P14780 1/20 0.52
USP2 O75604 1/20 0.52
PLAU P00749 1/20 0.52
HPN P05981 1/20 0.52
RAB9A P51151 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6151162 1.00 ITGA4 (0.58) ITGA4ITGB1ITGA2GAAHPGD
SCHEMBL6709564 0.91 ITGA4 (0.57) ITGA4ITGB1ITGA2GAAHPGD
SCHEMBL6710636 0.91 ITGA4 (0.57) ITGA4ITGB1ITGA2GAAHPGD
SCHEMBL6710949 0.90 GAA (0.60) ITGA4ITGB1ITGA2GAAHPGD
SCHEMBL5496192 0.89 ITGA4 (0.56) ITGA4ITGB1ITGA2GAAHPGD
SCHEMBL6709431 0.89 GAA (0.54) ITGA4ITGB1ITGA2GAAHPGD
SCHEMBL6714713 0.88 GAA (0.58) ITGA4ITGB1ITGA2GAAHPGD
SCHEMBL6714791 0.88 GAA (0.58) ITGA4ITGB1ITGA2GAAHPGD
SCHEMBL6400256 0.88 GAA (0.58) ITGA4ITGB1ITGA2GAAHPGD
SCHEMBL6400260 0.88 GAA (0.58) ITGA4ITGB1ITGA2GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1495044-A1 HETEROCYCLIC AMIDES WITH ALPHA-4 INTEGRIN ANTAGONIST ACTIVITY J. Uriach y Compania S.A. (ES) 2005-01-12 EP disclosed
WO-2003084984-A1 HETEROCYCLIC AMIDES WITH ALPHA-4 INTEGRIN ANTAGONIST ACTIVITY J. URIACH Y COMPANIA S.A. (ES) 2003-10-16 WO disclosed