Bromide

Bromide

SCHEMBL6151474

[Br-].c1ccc(N(c2ccccc2)[P+](N(c2ccccc2)c2ccccc2)(N(c2ccccc2)c2ccccc2)N(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHKA known ✓ P35790 4/20 0.34
ALDH1A1 P00352 8/20 0.38
NPSR1 Q6W5P4 2/20 0.38
ALOX15 P16050 1/20 0.38
HTT P42858 4/20 0.36
KMT2A Q03164 3/20 0.36
MAPT P10636 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
MEN1 O00255 2/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
HIF1A Q16665 1/20 0.35
HPGD P15428 2/20 0.33
GAA P10253 1/20 0.33
HSP90AA1 P07900 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7182773 0.94 ALDH1A1 (0.38) ALDH1A1NPSR1ALOX15HTTKMT2A
Bromide SCHEMBL6151384 0.69 ACHE (0.48) ALDH1A1HTTKMT2AMEN1TDP1
Bromide SCHEMBL28192148 0.67 ALDH1A1 (0.60) ALDH1A1NPSR1ALOX15HTTKMT2A
SCHEMBL453160 0.65 ALDH1A1 (0.67) ALDH1A1NPSR1ALOX15HTTKMT2A
SCHEMBL9490577 0.65 ALDH1A1 (0.67) ALDH1A1NPSR1ALOX15HTTKMT2A
Benzene SCHEMBL28083527 0.65 ALDH1A1 (0.67) ALDH1A1NPSR1ALOX15HTTKMT2A
SCHEMBL301494 0.65 ALDH1A1 (0.45) ALDH1A1NPSR1ALOX15HTTKMT2A
SCHEMBL30959 0.65 ALDH1A1 (0.67) ALDH1A1NPSR1ALOX15HTTKMT2A
SCHEMBL28366423 0.65 ALDH1A1 (0.39) ALDH1A1NPSR1ALOX15HTTKMT2A
SCHEMBL14570432 0.65 ALDH1A1 (0.39) ALDH1A1NPSR1ALOX15HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944564-B9 HALOGEN EXCHANGE REACTIONS AND USES THEREOF ALBEMARLE CORP (US) 2005-01-19 EP disclosed
EP-1054853-B1 CATALYST RECOVERY FOR HALOGEN EXCHANGE REACTIONS ALBEMARLE CORP (US) 2003-03-19 EP disclosed
US-6455718-B1 FOR CONTINUOUSLY RECOVERING CHLOROPENTAFLUOROBENZENE OR BROMOPENTAFLUOROBENZENE FROM VAPOR PHASE ALBEMARLE CORPORATION 2002-09-24 US disclosed
EP-0944564-B1 HALOGEN EXCHANGE REACTIONS AND USES THEREOF ALBEMARLE CORP (US) 2002-03-20 EP disclosed
US-6241917-B1 Halogen exchange reactions in preparing catalysts and their precursors ALBEMARLE CORPORATION 2001-06-05 US disclosed
US-6215032-B1 SOLVENT EXTRACTION; SEPARATING AMINOPHOSPHONIUM CATALYST; FLUORINATION OF HALOAROMATIC COMPOUND BY REPLACEMENT REACTION WITH ALKALI METAL FLUORIDE ALBEMARLE CORPORATION 2001-04-10 US disclosed
US-5965781-A PURIFYING THE CATALYST FOR IMPROVED PERFORMANCE BY DISSOLVING THE PHOSPHONIUM HALIDE IN A LIQUID CYCLIC ETHER, REMOVING THE SOLID IMPURITIES, ADDING A NONSOLVENT TO PRECIPITATE; REACTING AN ALKALI FLUORIDE AND HALO(S)BENZENE ALBEMARLE CORPORATION (US) 1999-10-12 US disclosed
US-5824827-A Halogen exchange reactions ALBEMARLE CORPORATION (US) 1998-10-20 US disclosed
US-5789631-A Production of perhalobenzenes ALBEMARLE CORPORATION (US) 1998-08-04 US disclosed