SCHEMBL6151773

SCHEMBL6151773

Cc1cn(-c2ccc(C(F)(F)F)cc2)nc1C

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.44
BRAF P15056 2/20 0.43
SRC P12931 1/20 0.43
KDR P35968 1/20 0.43
ADORA3 P0DMS8 2/20 0.42
KCNH2 Q12809 1/20 0.42
CTSS P25774 3/20 0.40
AADAT Q8N5Z0 1/20 0.40
PTGS2 P35354 2/20 0.40
CASR P41180 2/20 0.39
TDP1 Q9NUW8 1/20 0.37
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3060822 0.83 NOTUM (0.42) NOTUMBRAFSRCKDRADORA3
SCHEMBL17803164 0.82 NOTUM (0.52) NOTUMBRAFSRCKDRADORA3
SCHEMBL27497539 0.80 SRC (0.40) NOTUMBRAFSRCKDRADORA3
SCHEMBL19807433 0.80 KCNH2 (0.41) NOTUMBRAFSRCKDRADORA3
SCHEMBL17814158 0.80 CTSS (0.47) NOTUMBRAFSRCKDRADORA3
SCHEMBL27496521 0.80 SRC (0.40) NOTUMBRAFSRCKDRADORA3
SCHEMBL17973836 0.80 CTSS (0.47) NOTUMBRAFSRCKDRADORA3
SCHEMBL2611844 0.79 NPC1 (0.44) NOTUMBRAFSRCKDRADORA3
SCHEMBL5001181 0.79 NOTUM (0.52) NOTUMBRAFSRCKDRADORA3
SCHEMBL718415 0.79 PTGS2 (0.42) NOTUMBRAFSRCKDRADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106029640-B Pyrazolinone compounds and application thereof 泰普斯特医疗公司 2018-08-24 CN disclosed
EP-1585733-A1 HETEROCYCLIC PPAR MODULATORS ELI LILLY AND COMPANY (US) 2005-10-19 EP disclosed
WO-2004063166-A1 HETEROCYCLIC PPAR MODULATORS ELI LILLY AND COMPANY (US) 2004-07-29 WO disclosed