SCHEMBL6151897

SCHEMBL6151897

COc1ccc2c(C(=O)c3ccc(OCCC4CCCCN4)cc3)c(Cc3ccc(F)cc3)ccc2c1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.43
LTA4H P09960 5/20 0.39
CNR2 P34972 2/20 0.38
AURKB Q96GD4 1/20 0.38
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
NQO2 P16083 1/20 0.37
PTGER2 P43116 1/20 0.37
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
LTB4R Q15722 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6192190 0.87 CHEK2 (0.43) CHEK2ESR1ESR2NQO2
SCHEMBL6003394 0.85 CHEK2 (0.43) CHEK2LTA4HAURKBESR1ESR2
SCHEMBL6003300 0.84 CHEK2 (0.43) CHEK2LTA4HAURKBESR1ESR2
SCHEMBL6003307 0.84 CHEK2 (0.43) CHEK2LTA4HAURKBESR1ESR2
SCHEMBL5706403 0.84 CHEK2 (0.48) CHEK2LTA4HAURKBESR1ESR2
SCHEMBL5706380 0.84 CHEK2 (0.48) CHEK2LTA4HAURKBESR1ESR2
SCHEMBL6005363 0.83 CHEK2 (0.42) CHEK2LTA4HAURKBESR1ESR2
SCHEMBL6152202 0.83 LTA4H (0.39) CHEK2LTA4HAURKB
SCHEMBL6005756 0.83 CHEK2 (0.47) CHEK2LTA4HAURKBESR1ESR2
SCHEMBL6003358 0.83 CHEK2 (0.43) CHEK2LTA4HAURKBESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546139-A1 DERIVATIVE OF DIHYDRO-DIBENZO (A) ANTHRACENES AND THEIR USE AS SELECTIVE ESTROGEN RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 2005-06-29 EP disclosed
WO-2004029047-A1 DERIVATIVE OF DIHYDRO-DIBENZO (A) ANTHRACENES AND THEIR USE AS SELECTIVE ESTROGEN RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 2004-04-08 WO disclosed