SCHEMBL6151927

SCHEMBL6151927

Clc1ccc(C2(Cn3cncn3)COC(CBr)O2)c(Cl)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 15/20 0.62
CYP2C9 P11712 2/20 0.62
THRB P10828 1/20 0.53
KDM4E B2RXH2 1/20 0.44
LMNA P02545 2/20 0.40
FYN P06241 2/20 0.40
CYP51A1 Q16850 2/20 0.40
NR1I2 O75469 1/20 0.40
PGR P06401 1/20 0.40
HSP90AA1 P07900 1/20 0.40
CHRM2 P08172 1/20 0.40
CHRM4 P08173 1/20 0.40
CHRM5 P08912 1/20 0.40
ADRA2A P08913 1/20 0.40
CHRM1 P11229 1/20 0.40
TSHR P16473 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
CHRM3 P20309 1/20 0.40
DRD1 P21728 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6151930 1.00 CYP3A4 (0.62) CYP3A4CYP2C9THRBKDM4ELMNA
SCHEMBL9665341 0.86 CYP3A4 (0.46) CYP3A4CYP2C9THRBKDM4EHSP90AA1
SCHEMBL10517012 0.86 CYP3A4 (0.46) CYP3A4CYP2C9THRBKDM4EHSP90AA1
SCHEMBL74247 0.84 CYP3A4 (0.74) CYP3A4CYP2C9THRBKDM4ELMNA
SCHEMBL6152103 0.81 CYP3A4 (0.40) CYP3A4CYP2C9THRBLMNACYP51A1
SCHEMBL3046354 0.81 CYP3A4 (0.40) CYP3A4CYP2C9THRBLMNACYP51A1
SCHEMBL10518765 0.81 CYP3A4 (0.40) CYP3A4CYP2C9THRBLMNACYP51A1
SCHEMBL3046353 0.81 CYP3A4 (0.40) CYP3A4CYP2C9THRBLMNACYP51A1
SCHEMBL10516594 0.81 USP2 (0.45) CYP3A4CYP2C9LMNACYP51A1NR1I2
SCHEMBL9667152 0.81 USP2 (0.45) CYP3A4CYP2C9LMNACYP51A1NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1068200-B1 2,4,4-TRISUBSTITUTED-1,3-DIOXOLANE ANTIFUNGALS JANSSEN PHARMACEUTICA NV (BE) 2005-02-16 EP disclosed
US-6387906-B1 DERMATOPHYTES JANSSEN PHARMACEUTICA N.V. (BE) 2002-05-14 US disclosed