SCHEMBL6152206

SCHEMBL6152206

O=C(c1ccccc1-c1cccs1)N(Cc1ccc2ccccc2c1)C1Cc2ccccc2C1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 4/20 0.42
SLC6A4 P31645 4/20 0.42
SLC6A3 Q01959 3/20 0.42
MC4R P32245 1/20 0.42
MC5R P33032 1/20 0.42
MC3R P41968 1/20 0.42
KCNH2 Q12809 2/20 0.41
HCRTR1 O43613 12/20 0.40
HCRTR2 O43614 12/20 0.40
HTR1A P08908 2/20 0.36
HTR7 P34969 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5134499 0.88 HTR1A (0.40) HCRTR1HCRTR2HTR1AHTR7
SCHEMBL5135099 0.83 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3MC4RMC5R
SCHEMBL5137378 0.77 MC4R (0.45) SLC6A2SLC6A4SLC6A3MC4RMC5R
SCHEMBL5135649 0.74 C5AR1 (0.39)
SCHEMBL5136534 0.72 AGER (0.42)
SCHEMBL5137387 0.72 MEN1 (0.57) SLC6A2SLC6A4KCNH2
SCHEMBL5136513 0.72 TACR1 (0.43) SLC6A2SLC6A4KCNH2
SCHEMBL5137126 0.72 AGER (0.41)
SCHEMBL5135774 0.72 HSD17B2 (0.40) SLC6A2SLC6A4KCNH2
SCHEMBL5136654 0.70 MEN1 (0.49) SLC6A2SLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487796-A4 SUBSTITUTED BIARYL AMIDES AS C5A RECEPTOR MODULATORS NEUROGEN CORP (US) 2005-11-16 EP disclosed
EP-1487796-A1 SUBSTITUTED BIARYL AMIDES AS C5A RECEPTOR MODULATORS NEUROGEN CORPORATION (US) 2004-12-22 EP disclosed
WO-2003082826-A1 SUBSTITUTED BIARYL AMIDES AS C5A RECEPTOR MODULATORS NEUROGEN CORPORATION (US) 2003-10-09 WO disclosed