SCHEMBL6152239

SCHEMBL6152239

Clc1ccc(C2(Cn3ccnc3)COC(CBr)O2)cc1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HMOX1 P09601 2/20 0.42
CYP2A6 P11509 1/20 0.42
CYP19A1 P11511 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
CYP2B6 P20813 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6152242 1.00 HMOX1 (0.42) HMOX1CYP2A6CYP19A1CYP11B1CYP11B2
SCHEMBL27566787 0.91 HMOX1 (0.41) HMOX1CYP2A6CYP19A1CYP11B1CYP11B2
SCHEMBL6153207 0.90 CYP19A1 (0.40) HMOX1CYP19A1CYP11B1CYP11B2
SCHEMBL6153210 0.90 CYP19A1 (0.40) HMOX1CYP19A1CYP11B1CYP11B2
SCHEMBL10516594 0.86 USP2 (0.45) HMOX1CYP19A1CYP11B1CYP11B2
SCHEMBL9667152 0.86 USP2 (0.45) HMOX1CYP19A1CYP11B1CYP11B2
SCHEMBL27566788 0.81 HMOX1 (0.42) HMOX1CYP2A6CYP19A1CYP11B1CYP11B2
SCHEMBL27672581 0.81 CYP19A1 (0.39) HMOX1CYP19A1CYP11B1CYP11B2
SCHEMBL9665341 0.79 CYP3A4 (0.46)
SCHEMBL10517012 0.79 CYP3A4 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1068200-B1 2,4,4-TRISUBSTITUTED-1,3-DIOXOLANE ANTIFUNGALS JANSSEN PHARMACEUTICA NV (BE) 2005-02-16 EP disclosed
US-6387906-B1 DERMATOPHYTES JANSSEN PHARMACEUTICA N.V. (BE) 2002-05-14 US disclosed