SCHEMBL6152270

SCHEMBL6152270

O=c1oc2cc(O)ccc2c(Cc2ccc(OCCC3CCCN3)cc2)c1-c1ccc(C(F)(F)F)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 17/20 0.47
ESR2 Q92731 3/20 0.44
AR P10275 1/20 0.38
HSD17B3 P37058 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6152455 0.91 CYP19A1 (0.44) ESR1
SCHEMBL5983904 0.90 ESR1 (0.48) ESR1ESR2
SCHEMBL4640167 0.89 ESR1 (0.57) ESR1ESR2
SCHEMBL6158194 0.88 ESR1 (0.45) ESR1ESR2ARHSD17B3
SCHEMBL5416855 0.86 ESR1 (0.54) ESR1ESR2
SCHEMBL4619222 0.85 ESR1 (0.55) ESR1ESR2
SCHEMBL6153596 0.81 CYP19A1 (0.51) ESR1ESR2
SCHEMBL4641971 0.81 ESR1 (0.59) ESR1ESR2
SCHEMBL6152326 0.80 CYP19A1 (0.51) ESR1
SCHEMBL4621568 0.79 ESR1 (0.55) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1497277-A1 BENZOPYRANONE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH Signal Pharmaceuticals, Inc. (US) 2005-01-19 EP disclosed
WO-2003089422-A1 BENZOPYRANONE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH SIGNAL PHARMACEUTICALS, INC. (US) 2003-10-30 WO disclosed