SCHEMBL6152326

SCHEMBL6152326

COc1ccc2c(Cc3ccc(OCCC4CCCN4)cc3)c(-c3ccc(C(F)(F)F)cc3)c(=O)oc2c1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.51
ESR1 P03372 10/20 0.51
DRD2 P14416 1/20 0.45
DRD4 P21917 1/20 0.45
DRD3 P35462 1/20 0.45
MAOB P27338 1/20 0.43
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4640167 0.91 ESR1 (0.57) ESR1
SCHEMBL4639556 0.90 ESR1 (0.42) CYP19A1ESR1DRD2DRD4DRD3
SCHEMBL4639606 0.90 ESR1 (0.41) CYP19A1ESR1DRD2DRD4DRD3
SCHEMBL4639760 0.89 ESR1 (0.45) CYP19A1ESR1
SCHEMBL6152455 0.89 CYP19A1 (0.44) CYP19A1ESR1DRD2DRD4DRD3
SCHEMBL4640636 0.86 ESR1 (0.45) ESR1
SCHEMBL5422253 0.85 ESR1 (0.64) CYP19A1ESR1DRD2DRD4DRD3
SCHEMBL6153596 0.81 CYP19A1 (0.51) CYP19A1ESR1DRD2DRD4DRD3
SCHEMBL4640144 0.81 ESR1 (0.64) CYP19A1ESR1DRD2DRD4DRD3
SCHEMBL4639650 0.80 ESR1 (0.42) ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1497277-A1 BENZOPYRANONE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH Signal Pharmaceuticals, Inc. (US) 2005-01-19 EP disclosed
WO-2003089422-A1 BENZOPYRANONE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH SIGNAL PHARMACEUTICALS, INC. (US) 2003-10-30 WO disclosed