SCHEMBL6152826

SCHEMBL6152826

Cc1cc([C@H]2C[C@@H]3CC[C@H]([C@H]2CCl)N3C)ccc1Cl

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 14/20 0.62
SLC6A4 P31645 13/20 0.62
SLC6A2 P23975 8/20 0.62
CHRNA1 P02708 4/20 0.60
CHRNG P07510 4/20 0.60
ITGA5 P08648 4/20 0.60
CHRNB1 P11230 4/20 0.60
CHRNB2 P17787 4/20 0.60
CHRNB4 P30926 4/20 0.60
CHRNA3 P32297 4/20 0.60
CHRNA4 P43681 4/20 0.60
CHRND Q07001 4/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6152828 1.00 SLC6A3 (0.62) SLC6A3SLC6A4SLC6A2CHRNA1CHRNG
SCHEMBL6152899 0.90 SLC6A3 (0.76) SLC6A3SLC6A4SLC6A2
SCHEMBL6152901 0.90 SLC6A3 (0.76) SLC6A3SLC6A4SLC6A2
SCHEMBL8291598 0.85 SLC6A3 (0.83) SLC6A3SLC6A4SLC6A2CHRNA1CHRNG
SCHEMBL14173845 0.83 SLC6A3 (0.82) SLC6A3SLC6A4SLC6A2
SCHEMBL5731247 0.83 SLC6A3 (0.82) SLC6A3SLC6A4SLC6A2
SCHEMBL5731249 0.83 SLC6A3 (0.82) SLC6A3SLC6A4SLC6A2
SCHEMBL6574444 0.79 SLC6A3 (0.74) SLC6A3SLC6A4SLC6A2
SCHEMBL6574468 0.79 SLC6A3 (0.74) SLC6A3SLC6A4SLC6A2
SCHEMBL7343838 0.79 SLC6A3 (0.74) SLC6A3SLC6A4SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0897922-B1 Cocaine receptor binding ligands RES TRIANGLE INST (US) 2005-07-20 EP disclosed
EP-0897922-A2 Cocaine receptor binding ligands RESEARCH TRIANGLE INSTITUTE (US) 1999-02-24 EP disclosed
US-5736123-A TRIALKYLTIN CHEMICAL INTERMEDIATES RESEARCH TRIANGLE INSTITUTE (US) 1998-04-07 US disclosed
US-5496953-A DOPAMINE TRANSPORTER SITES, RADIOACTIVE, DIAGNOSIS, IMAGING, NORTROPANE DERIVATIVES RESEARCH TRIANGLE INSTITUTE (US) 1996-03-05 US disclosed
US-5380848-A 8-azabicyclo(3.2.1)octanes RESEARCH TRIANGLE INSTITUTE (US) 1995-01-10 US disclosed
WO-1993009814-A1 COCAINE RECEPTOR BINDING LIGANDS RESEARCH TRIANGLE INSTITUTE (US) 1993-05-27 WO disclosed