SCHEMBL6152840

SCHEMBL6152840

COc1ccc2c(C(=O)c3ccc(OCCC4CCCCN4)cc3)c(Cc3ccccc3)sc2c1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 14/20 0.49
ESR2 Q92731 14/20 0.49
LTA4H P09960 2/20 0.43
CHEK2 O96017 1/20 0.43
CNR2 P34972 3/20 0.42
CNR1 P21554 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6197784 0.90 ESR1 (0.45) ESR1ESR2CHEK2CNR2CNR1
SCHEMBL6773068 0.84 ESR1 (0.66) ESR1ESR2CNR2CNR1
SCHEMBL6204005 0.83 ESR1 (0.49) ESR1ESR2CHEK2
SCHEMBL6153041 0.83 ESR1 (0.49) ESR1ESR2CHEK2
Hydrochloric Acid SCHEMBL6767144 0.83 ESR1 (0.67) ESR1ESR2CNR1
SCHEMBL6152532 0.83 LTA4H (0.43) LTA4HCHEK2
SCHEMBL5826488 0.81 ESR1 (0.73) ESR1ESR2
SCHEMBL6195029 0.81 ESR1 (0.53) ESR1ESR2CNR1
SCHEMBL7817127 0.81 CNR2 (0.61) ESR1ESR2CNR2CNR1
SCHEMBL5706945 0.80 ESR1 (0.51) ESR1ESR2CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546139-A1 DERIVATIVE OF DIHYDRO-DIBENZO (A) ANTHRACENES AND THEIR USE AS SELECTIVE ESTROGEN RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 2005-06-29 EP claimed
WO-2004029047-A1 DERIVATIVE OF DIHYDRO-DIBENZO (A) ANTHRACENES AND THEIR USE AS SELECTIVE ESTROGEN RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 2004-04-08 WO claimed
EP-1546139-A1 DERIVATIVE OF DIHYDRO-DIBENZO (A) ANTHRACENES AND THEIR USE AS SELECTIVE ESTROGEN RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 2005-06-29 EP disclosed
WO-2004029047-A1 DERIVATIVE OF DIHYDRO-DIBENZO (A) ANTHRACENES AND THEIR USE AS SELECTIVE ESTROGEN RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 2004-04-08 WO disclosed