SCHEMBL6153041

SCHEMBL6153041

COc1ccc2c(C(=O)c3ccc(OCCC4CCCCN4)cc3)c(N(C)C)sc2c1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 15/20 0.49
ESR2 Q92731 15/20 0.49
CHEK2 O96017 1/20 0.44
ENPP1 P22413 2/20 0.43
ENPP3 O14638 2/20 0.42
AURKB Q96GD4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6773068 0.87 ESR1 (0.66) ESR1ESR2ENPP1ENPP3
Hydrochloric Acid SCHEMBL6767144 0.86 ESR1 (0.67) ESR1ESR2ENPP1ENPP3
SCHEMBL6152840 0.83 ESR1 (0.49) ESR1ESR2CHEK2
SCHEMBL6197784 0.81 ESR1 (0.45) ESR1ESR2CHEK2ENPP1ENPP3
SCHEMBL6204005 0.81 ESR1 (0.49) ESR1ESR2CHEK2ENPP1ENPP3
SCHEMBL4818774 0.80 ESR1 (0.75) ESR1ESR2ENPP1ENPP3
Hydrochloric Acid SCHEMBL9271052 0.79 ESR1 (0.75) ESR1ESR2ENPP1ENPP3
SCHEMBL5706403 0.78 CHEK2 (0.48) ESR1ESR2CHEK2AURKB
SCHEMBL5706380 0.78 CHEK2 (0.48) ESR1ESR2CHEK2AURKB
SCHEMBL5706945 0.78 ESR1 (0.51) ESR1ESR2CHEK2ENPP1ENPP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1551822-A2 PENTACYCLIC OXEPINES AND DERIVATIVES THEREOF, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ELI LILLY AND COMPANY (US) 2005-07-13 EP disclosed
EP-1546139-A1 DERIVATIVE OF DIHYDRO-DIBENZO (A) ANTHRACENES AND THEIR USE AS SELECTIVE ESTROGEN RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 2005-06-29 EP disclosed
EP-1527076-A1 DIHYDRO-DIBENZO (B,E) OXEPINE BASED SELECTIVE ESTROGEN RECEPTOR MODULATORS, COMPOSITIONS AND METHODS ELI LILLY AND COMPANY (US) 2005-05-04 EP disclosed
WO-2004029047-A1 DERIVATIVE OF DIHYDRO-DIBENZO (A) ANTHRACENES AND THEIR USE AS SELECTIVE ESTROGEN RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 2004-04-08 WO disclosed
WO-2004009578-A2 PENTACYCLIC OXEPINES AND DERIVATIVES THEREOF, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ELI LILLY AND COMPANY (US) 2004-01-29 WO disclosed
WO-2004009603-A1 DIHYDRO-DIBENZO[B,E]OXEPINE BASED SELECTIVE ESTROGEN RECEPTOR MODULATORS, COMPOSITIONS AND METHODS ELI LILLY AND COMPANY (US) 2004-01-29 WO disclosed