SCHEMBL6152875

SCHEMBL6152875

O=C(C=Cc1ccccc1)Nc1ccc2[nH]nnc2c1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.57
MMP1 P03956 9/20 0.55
MMP2 P08253 9/20 0.55
MMP9 P14780 9/20 0.55
EGFR P00533 9/20 0.55
MAOA P21397 4/20 0.55
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
ALDH1A1 P00352 2/20 0.54
MAPT P10636 2/20 0.54
KDM4E B2RXH2 1/20 0.54
DEGS1 O15121 1/20 0.53
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
TOP2A P11388 1/20 0.51
POLB P06746 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
CA12 O43570 1/20 0.51
CA9 Q16790 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6152873 1.00 MAOB (0.57) MAOBMMP1MMP2MMP9EGFR
SCHEMBL13675670 0.85 TRPV1 (0.61) MEN1KMT2AMAPTKDM4ENPC1
SCHEMBL9506585 0.84 ALDH1A1 (0.58) KMT2AALDH1A1MAPTKDM4EPOLB
SCHEMBL9876497 0.84 ALDH1A1 (0.58) KMT2AALDH1A1MAPTKDM4EPOLB
SCHEMBL10949559 0.79 MAP2K7 (0.45) EGFR
SCHEMBL9474776 0.79 KDM4E (0.40) MAOBEGFRMAOAKMT2AALDH1A1
SCHEMBL9474772 0.79 KDM4E (0.40) MAOBEGFRMAOAKMT2AALDH1A1
SCHEMBL7773324 0.78 NPC1 (0.59) MAOBMAOAMEN1KMT2AALDH1A1
SCHEMBL8767799 0.77 MMP2 (0.61) MAOBMMP1MMP2MMP9EGFR
SCHEMBL13836663 0.77 MMP2 (0.61) MAOBMMP1MMP2MMP9EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 42 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-H963-H Containing development inhibitor and reducible dye FUJI PHOTO FILM CO., LTD. (JP) 1991-09-03 US claimed
EP-1037106-B1 Color diffusion transfer photographic material FUJI PHOTO FILM CO LTD (JP) 2005-01-26 EP disclosed
US-6376164-B1 CONTAINING 2-THIOBENZOTHIAZOLE COMPOUND FUJI PHOTO FILM CO., LTD. (JP) 2002-04-23 US disclosed
US-6187527-B1 A SENSITIVITY REGULATION BY PROLONGING THE BLACK AND WHITE DEVELOPMENT TIME DURING COLOR REVERSAL PROCESS IS CONDUCTED IN ORDER TO COMPENSATE FOR ANY UNDER-EXPOSURE OF A COLOR PHOTOGRAPHIC LIGHTSENSITIVE MATERIAL. FUJI PHOTO FILM CO., LTD. (JP) 2001-02-13 US disclosed
EP-1037106-A1 Color diffusion transfer photographic material FUJI PHOTO FILM CO., LTD. (JP) 2000-09-20 EP disclosed
US-6013421-A EXPOSURE TO LIGHT FOR SILVER HALIDE EMULSIONS FOR COLOR PHOTOGRAPHY FUJI PHOTO FILM CO., LTD. (JP) 2000-01-11 US disclosed
EP-0534283-B1 Silver halide photographic light-sensitive material FUJI PHOTO FILM CO LTD (JP) 1997-12-17 EP disclosed
US-5691125-A CYAN DYE-FORMING COUPLER, STORAGE STABLE FUJI PHOTO FILM CO., LTD. (JP) 1997-11-25 US disclosed
US-5609999-A INDOLE DYE; STORAGE STABILITY, COLOR REPRODUCIBILITY, SHARPNESS FUJI PHOTO FILM CO., LTD. (JP) 1997-03-11 US disclosed
EP-0537659-B1 Silver halide color photographic light-sensitive material, and method of processing the same FUJI PHOTO FILM CO LTD (JP) 1997-01-15 EP disclosed
US-4939066-A DEVELOPMENT INHIBITOR-RELEASING COMPOUND FUJI PHOTO FILM CO., LTD. (JP) 1990-07-03 US disclosed
US-4891304-A RELEASE OF PHOTOGRAPHICALLY USEFUL COMPOUND BY REDUCTIVE CLEAVAGE OF NITROGEN-NITROGEN BOND FUJI PHOTO FILM CO., LTD. (JP) 1990-01-02 US disclosed
US-4886736-A COUPLERS AND COMPOUND CAPABLE OF RELEASING PHOTOGRAPHICALLY USEFUL GROUP UPON REDUCTION FUJI PHOTO FILM CO., LTD. (JP) 1989-12-12 US disclosed
EP-0198438-B1 SILVER HALIDE PHOTOGRAPHIC LIGHT-SENSITIVE MATERIAL FUJI PHOTO FILM CO., LTD. (JP) 1989-10-18 EP disclosed
US-4840887-A USEFUL GROUP RELEASED BY CLEAVAGE BETWEEN SULFONYL GROUP AND A NITROGEN, SULFUR OR OXYGEN ATOM; STABILITY FUJI PHOTO FILM CO., LTD. (JP) 1989-06-20 US disclosed
US-4820622-A RELEASING DIFFUSIBLE DYE IN ALKALINE SYSTEM AFTER HALIDE REDUCTION FUJI PHOTO FILM CO., LTD. (JP) 1989-04-11 US disclosed
US-4783396-A Silver halide photographic materials FUJI PHOTO FILM CO., LTD. (JP) 1988-11-08 US disclosed
US-4770990-A Silver halide photographic light-sensitive material containing a compound capable of imagewise releasing a photographically useful group during development FUJI PHOTO FILM CO., LTD. (JP) 1988-09-13 US disclosed
EP-0220746-A2 Silver halide photographic materials FUJI PHOTO FILM CO., LTD. (JP) 1987-05-06 EP disclosed
EP-0198438-A2 Silver halide photographic light-sensitive material FUJI PHOTO FILM CO., LTD. (JP) 1986-10-22 EP disclosed