SCHEMBL6153084

SCHEMBL6153084

CC1(c2ccc3c(c2)OCO3)CC(Nc2n[nH]cc2C(=O)O)C(=O)O1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.36
GAA P10253 2/20 0.35
CFTR P13569 2/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
ALDH1A1 P00352 2/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CRHBP P24387 1/20 0.34
CRHR2 Q13324 1/20 0.34
MAPK1 P28482 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6152278 0.89 ALDH1A1 (0.45) CFTRMAPTALDH1A1SMN1; SMN2MAPK1
SCHEMBL6153355 0.85
SCHEMBL6152990 0.83 NPC1 (0.33) CYP2C9GAAMAPTHTTALDH1A1
SCHEMBL6153162 0.83 ALDH1A1 (0.40) CYP2C9CFTRMAPTHTTALDH1A1
SCHEMBL6295391 0.80 CYP2C9 (0.34) CYP2C9GAAMAPTHTTALDH1A1
SCHEMBL6152459 0.77 NPC1 (0.49) CYP2C9GAACFTRMAPTHTT
SCHEMBL6152267 0.74 NPC1 (0.47) GAAMAPTHTTALDH1A1SMN1; SMN2
SCHEMBL6152274 0.74 MAPT (0.46) GAACFTRMAPTHTTALDH1A1
SCHEMBL6291829 0.74 JAK2 (0.40) GAAMAPTALDH1A1SMN1; SMN2MEN1
SCHEMBL6152524 0.72 CRHBP (0.41) GAACFTRMAPTHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1406610-B1 USE OF SUBSTITUTED GAMMA-LACTONE COMPOUNDS AS MEDICAMENTS GRUENENTHAL GMBH (DE) 2005-01-26 EP claimed