SCHEMBL6154372

SCHEMBL6154372

COc1cccc(Oc2cc(Oc3cccc(OC)c3)cc(-c3nnc(Nc4cccc(C(=O)O)c4)s3)c2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.53
RAB9A P51151 4/20 0.53
GSK3B P49841 1/20 0.51
MITF O75030 1/20 0.50
AKR1C3 P42330 2/20 0.49
AKR1C2 P52895 2/20 0.49
DYRK1A Q13627 1/20 0.48
ROCK2 O75116 1/20 0.48
ROCK1 Q13464 1/20 0.48
CSNK2A1 P68400 2/20 0.48
FABP1 P07148 1/20 0.48
KDM4E B2RXH2 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
ALDH1A1 P00352 2/20 0.47
USP2 O75604 1/20 0.47
HPGD P15428 1/20 0.47
HSD17B10 Q99714 1/20 0.47
MAPK13 O15264 1/20 0.47
MAPK12 P53778 1/20 0.47
MAPK11 Q15759 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5558657 0.88 NPC1 (0.53) NPC1RAB9AAKR1C3AKR1C2DYRK1A
SCHEMBL6153554 0.86 AKR1C3 (0.47) AKR1C3AKR1C2ROCK2ROCK1KDM4E
SCHEMBL5556608 0.81 ROCK2 (0.50) NPC1RAB9AAKR1C3AKR1C2ROCK2
SCHEMBL5556693 0.81 ROCK1 (0.49) NPC1RAB9AGSK3BDYRK1AROCK2
SCHEMBL6154251 0.79 NR1H4 (0.54) NPC1RAB9AROCK2ROCK1MEN1
SCHEMBL6153810 0.78 KMO (0.55) NPC1RAB9AAKR1C3ROCK2ROCK1
SCHEMBL5464421 0.75 NPC1 (0.78) NPC1RAB9AGSK3BMITFAKR1C3
SCHEMBL6244318 0.74 SMN1; SMN2 (0.47) NPC1RAB9ADYRK1AROCK1CSNK2A1
SCHEMBL5556610 0.74 AKR1C3 (0.44) NPC1RAB9AAKR1C3AKR1C2ROCK2
SCHEMBL2867923 0.74 AKR1C3 (0.73) NPC1RAB9AMITFAKR1C3FABP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050065118-A1 Organosulfur inhibitors of tyrosine phosphatases METABASIS THERAPEUTICS, INC. 2005-03-24 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050065118-A1 Organosulfur inhibitors of tyrosine phosphatases PTPRS, PTPRJ, PTPRCAP NPC1 4548/4885RAB9A 3814/4885GSK3B 3097/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.