Isothiocyanate

Isothiocyanate

SCHEMBL6154717

Brc1ccccc1Br.N=C=S

nearest known ligand 0.41

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
MAPK1 P28482 2/20 0.38
TDP1 Q9NUW8 2/20 0.35
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA4 P22748 1/20 0.35
CA6 P23280 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
TAAR1 Q96RJ0 3/20 0.33
GAA P10253 2/20 0.33
CA5A P35218 1/20 0.32
CA9 Q16790 1/20 0.32
IDO1 P14902 2/20 0.32
PLCG1 P19174 1/20 0.32
MIF P14174 1/20 0.32
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
MPI P34949 1/20 0.31
DCUN1D1 Q96GG9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Isothiocyanate SCHEMBL6154362 0.82 TSHR (0.41) ALDH1A1MAPK1GAAMAPTHSD11B1
Isothiocyanate SCHEMBL2893068 0.82 HTT (0.37) ALDH1A1MAPK1TDP1CA1CA2
Isothiocyanate SCHEMBL2886977 0.82 ALDH1A1 (0.71) ALDH1A1MAPK1TDP1CA1CA2
SCHEMBL29314 0.79
SCHEMBL29404525 0.79
Bromobenzene SCHEMBL6154095 0.79 ALDH1A1 (0.65) ALDH1A1MAPK1TDP1MIFKDM4E
Isothiocyanate SCHEMBL27973971 0.78 CA2 (0.46) ALDH1A1TDP1CA1CA2L3MBTL1
SCHEMBL9651341 0.75
SCHEMBL30007372 0.75
Lithium SCHEMBL9651351 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050065118-A1 Organosulfur inhibitors of tyrosine phosphatases METABASIS THERAPEUTICS, INC. 2005-03-24 US disclosed
EP-1446110-A2 ORGANOSULFUR INHIBITORS OF TYROSINE PHOSPHATASES Structural Bioinformatics Inc. (US) 2004-08-18 EP disclosed
WO-2003032916-A2 ORGANOSULFUR INHIBITORS OF TYROSINE PHOSPHATASES STRUCTURAL BIOINFORMATICS INC. (US) 2003-04-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050065118-A1 Organosulfur inhibitors of tyrosine phosphatases PTPRS, PTPRJ, PTPRCAP ALDH1A1 961/4885MAPK1 2027/4885TDP1 219/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.