SCHEMBL6154730

SCHEMBL6154730

O=C(O)CC(c1c[c]ccc1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 1/20 0.45
CACNA1B Q00975 1/20 0.45
CACNB1 Q02641 1/20 0.45
CACNA1C Q13936 1/20 0.45
ACP3 P15309 2/20 0.44
CES2 O00748 1/20 0.44
PNMT P11086 1/20 0.43
SLC6A9 P48067 2/20 0.42
FFAR1 O14842 1/20 0.42
CTSA P10619 4/20 0.41
TACR1 P25103 1/20 0.41
EPHX1 P07099 2/20 0.40
BCHE P06276 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
POLB P06746 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6153911 0.85 ALDH1A1 (0.41) CACNA2D1CACNA1BCACNB1CACNA1CACP3
Hydrochloric Acid SCHEMBL9293074 0.83 CACNA2D1 (0.56) CACNA2D1CACNA1BCACNB1CACNA1CACP3
SCHEMBL6153418 0.80 GAA (0.44) CACNA2D1CACNA1BCACNB1CACNA1CACP3
SCHEMBL6156534 0.78 EPHX1 (0.41) ACP3CES2PNMTSLC6A9FFAR1
SCHEMBL6155403 0.77 PNMT (0.50) ACP3CES2PNMTALDH1A1
SCHEMBL5856970 0.77 PNMT (0.53) CACNA2D1CACNA1BCACNB1CACNA1CACP3
SCHEMBL23125123 0.75 ACP3 (0.50) CACNA2D1CACNA1BCACNB1CACNA1CACP3
SCHEMBL11336248 0.75 ACP3 (0.50) CACNA2D1CACNA1BCACNB1CACNA1CACP3
SCHEMBL4730061 0.75 ACP3 (0.50) CACNA2D1CACNA1BCACNB1CACNA1CACP3
SCHEMBL382119 0.75 PNMT (0.54) CACNA2D1CACNA1BCACNB1CACNA1CACP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050065118-A1 Organosulfur inhibitors of tyrosine phosphatases METABASIS THERAPEUTICS, INC. 2005-03-24 US disclosed
EP-1446110-A2 ORGANOSULFUR INHIBITORS OF TYROSINE PHOSPHATASES Structural Bioinformatics Inc. (US) 2004-08-18 EP disclosed
WO-2003032916-A2 ORGANOSULFUR INHIBITORS OF TYROSINE PHOSPHATASES STRUCTURAL BIOINFORMATICS INC. (US) 2003-04-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050065118-A1 Organosulfur inhibitors of tyrosine phosphatases PTPRS, PTPRJ, PTPRCAP CACNA2D1 3781/4885CACNA1B 3775/4885CACNB1 3320/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.