SCHEMBL6155937

SCHEMBL6155937

Cc1ncn(Cc2ccccc2)c2nc(N)nc1-2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.49
ADORA1 P30542 2/20 0.49
CYP1A2 P05177 2/20 0.49
ALDH1A1 P00352 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
HIF1A Q16665 1/20 0.49
PHLPP2 Q6ZVD8 1/20 0.49
LMNA P02545 1/20 0.46
FLT1 P17948 1/20 0.45
KDR P35968 1/20 0.45
TEK Q02763 1/20 0.45
HRH4 Q9H3N8 1/20 0.45
PI4KA P42356 1/20 0.43
PI4K2B Q8TCG2 1/20 0.43
PI4K2A Q9BTU6 1/20 0.43
PI4KB Q9UBF8 1/20 0.43
TNF P01375 1/20 0.43
CYP11B1 P15538 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6155911 0.83 ADORA2A (0.48) ADORA2AADORA1CYP1A2ALDH1A1CYP3A4
SCHEMBL22598664 0.77 ADORA2A (0.47) ADORA2AADORA1CYP1A2ALDH1A1CYP3A4
SCHEMBL2566348 0.74 CYP11B1 (0.53) ADORA2AALDH1A1LMNAPI4KAPI4K2B
SCHEMBL22598712 0.71 ADORA2A (0.48) ADORA2AADORA1ALDH1A1LMNAFLT1
SCHEMBL25543494 0.71 ADORA2A (0.70) ADORA2AADORA1CYP1A2ALDH1A1CYP3A4
SCHEMBL21199068 0.71 ADORA2A (0.54) ADORA2ALMNAPI4KAPI4K2BPI4K2A
3-Benzyladenine SCHEMBL5352368 0.70 ADORA2A (0.56) ADORA2AALDH1A1LMNAPI4KAPI4K2B
SCHEMBL11211782 0.69 CYP11B1 (0.47) ADORA2ALMNAPI4KAPI4K2BPI4K2A
Hydrochloric Acid SCHEMBL11295371 0.69 CYP11B1 (0.47) ADORA2AALDH1A1LMNAPI4KAPI4K2B
SCHEMBL1640041 0.69 PDE4A (0.69) ADORA2AADORA1CYP1A2ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0912575-B1 PROCESSES FOR THE SYNTHESIS OF CHEMICAL COMPOUNDS HAVING PDE-IV INHIBITORY ACTIVITY EURO CELTIQUE SA (LU) 2005-02-02 EP disclosed
US-6310205-B1 Hypoxathine compounds EURO-CELTIQUE, S.A. (LU) 2001-10-30 US disclosed
EP-0912575-A4 IMPROVED METHODS FOR THE SYNTHESIS OF CHEMICAL COMPOUNDS HAVING PDE-IV INHIBITORY ACTIVITY EURO CELTIQUE SA (LU) 2001-04-25 EP disclosed
EP-0912575-A1 IMPROVED METHODS FOR THE SYNTHESIS OF CHEMICAL COMPOUNDS HAVING PDE-IV INHIBITORY ACTIVITY Euro-Celtique S.A. (LU) 1999-05-06 EP disclosed
US-5864037-A Methods for the synthesis of chemical compounds having PDE-IV inhibitory activity EURO-CELTIQUE, S.A. (LU) 1999-01-26 US disclosed
WO-1997046561-A1 IMPROVED METHODS FOR THE SYNTHESIS OF CHEMICAL COMPOUNDS HAVING PDE-IV INHIBITORY ACTIVITY EURO-CELTIQUE, S.A. (LU) 1997-12-11 WO disclosed