SCHEMBL6155985

SCHEMBL6155985

Cc1cc(CC=O)cc(Cl)c1N

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CD44 P16070 1/20 0.35
CYP1A1 P04798 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 4/20 0.34
ALDH1A1 P00352 3/20 0.34
TP53 P04637 1/20 0.34
TSHR P16473 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
POLB P06746 1/20 0.30
ATP4A P20648 1/20 0.30
ATP4B P51164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5746917 0.87 ALDH1A1 (0.46) CYP3A4ALDH1A1TSHRTDP1CA1
SCHEMBL7642936 0.81 CYP3A4 (0.45) CD44CYP1A1CYP1A2CYP3A4ALDH1A1
SCHEMBL30806137 0.81 CYP3A4 (0.45) CD44CYP1A1CYP1A2CYP3A4ALDH1A1
SCHEMBL11139083 0.79 CD44 (0.38) CD44CYP1A1CYP1A2CYP3A4ALDH1A1
SCHEMBL2003716 0.79 CD44 (0.38) CD44CYP1A1CYP1A2CYP3A4ALDH1A1
SCHEMBL3410728 0.73 MCL1 (0.40) ALDH1A1TSHRPOLB
SCHEMBL7044076 0.73 ALDH1A1 (0.44) CYP3A4ALDH1A1POLB
SCHEMBL8756021 0.73 ALDH1A1 (0.41) CYP3A4ALDH1A1TSHRTDP1
SCHEMBL25261330 0.73 ATP4A (0.45) CYP1A1CYP1A2CYP3A4ALDH1A1TP53
SCHEMBL21603385 0.73 CYP3A4 (0.37) CD44CYP1A1CYP1A2CYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1597242-A1 HIV INHIBITING 1,2,4-TRIAZINES JANSSEN PHARMACEUTICA N.V. (BE) 2005-11-23 EP disclosed
EP-0940139-B1 Substituted guanidines and derivatives thereof as modulators of neurotransmitter release and novel methodology for identifying neurotransmitter release blockers SCION PHARMACEUTICALS INC (US) 2005-02-02 EP disclosed
WO-2004074266-A1 HIV INHIBITING 1,2,4-TRIAZINES JANSSEN PHARMACEUTICA N.V. (BE) 2004-09-02 WO disclosed
US-5637623-A CENTRAL NERVOUS SYSTEM DISORDERS CAMBRIDGE NEUROSCIENCE, INC. (US) 1997-06-10 US disclosed