SCHEMBL6156448

SCHEMBL6156448

Cc1c(O)ccc2c(N3CCOCC3)cc(=O)oc12

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 10/20 0.64
MAOB P27338 1/20 0.57
PDE3B Q13370 1/20 0.53
PDE3A Q14432 1/20 0.53
CASP1 P29466 1/20 0.52
CASP7 P55210 1/20 0.52
HSD17B10 Q99714 1/20 0.52
CA12 O43570 2/20 0.50
CA9 Q16790 2/20 0.50
TNF P01375 1/20 0.50
NOD2 Q9HC29 1/20 0.50
NOD1 Q9Y239 1/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
GLA P06280 1/20 0.50
P4HB P07237 1/20 0.50
GAA P10253 1/20 0.50
HPGD P15428 1/20 0.50
KMT2A Q03164 1/20 0.48
ATM Q13315 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6155892 0.88 MAOB (0.58) PRKDCMAOBCA12CA9TNF
SCHEMBL6156974 0.84 ERAP1 (0.58) PRKDCMAOBPDE3BPDE3ACA12
SCHEMBL6155495 0.82 MAOB (0.51) PRKDCMAOBPDE3BPDE3ACA12
SCHEMBL7321820 0.79 P2RY12 (0.70) PRKDC
SCHEMBL31060159 0.78 PRKDC (1.00) PRKDC
SCHEMBL7317237 0.77 P2RY12 (0.60) MAOBCASP1CASP7HSD17B10KDM4E
SCHEMBL5345045 0.75 MAOB (0.77) MAOBCA12CA9TNFNOD2
SCHEMBL31060570 0.75 PRKDC (1.00) PRKDC
SCHEMBL28365890 0.74 KMT2A (0.62) PRKDCPDE3BPDE3AHSD17B10KDM4E
SCHEMBL28499055 0.74 PRKDC (0.68) PRKDCMAOBCASP1CASP7HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894805-B1 Ribose substituted aromatic derivatives, their preparation and use as medicaments AVENTIS PHARMA SA (FR) 2005-02-09 EP disclosed
US-5968939-A ANTIBIOTICS FROM AMINOOXOBENZOPYRAN COMPOUNDS HOECHST MARION ROUSSEL (FR) 1999-10-19 US disclosed
EP-0894805-A1 Ribose substituted aromatic derivatives, their preparation and use as medicaments HOECHST MARION ROUSSEL (FR) 1999-02-03 EP disclosed