SCHEMBL6157322

SCHEMBL6157322

Cc1c(O)ccc2c(N3CCN(C)CC3)c(Cl)c(=O)oc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERAP1 Q9NZ08 1/20 0.52
CCR4 P51679 4/20 0.50
ESR2 Q92731 6/20 0.48
ESR1 P03372 5/20 0.48
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 3/20 0.47
GAA P10253 3/20 0.47
GLA P06280 2/20 0.47
HPGD P15428 2/20 0.47
MAOA P21397 1/20 0.47
MAPK1 P28482 1/20 0.47
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
HSD17B10 Q99714 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MAOB P27338 1/20 0.45
MAPT P10636 1/20 0.44
HIF1A Q16665 1/20 0.44
CA12 O43570 1/20 0.43
CA9 Q16790 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9211529 0.76 KDM4E (0.66) ESR2ESR1KDM4EALDH1A1GAA
SCHEMBL16260714 0.75 MAOB (0.48) ERAP1CCR4ESR2ESR1KDM4E
SCHEMBL6155892 0.75 MAOB (0.58) ERAP1CCR4KDM4EALDH1A1GAA
Hydrochloric Acid SCHEMBL16242701 0.74 MAOB (0.47) ERAP1CCR4ESR2ESR1KDM4E
SCHEMBL3766383 0.70 KDM4E (0.74) ESR2ESR1KDM4EALDH1A1GAA
SCHEMBL27806711 0.67 CCR4 (1.00) CCR4
SCHEMBL28065504 0.66 ESR2 (0.56) ERAP1ESR2ESR1KDM4EALDH1A1
SCHEMBL6828759 0.66 ESR2 (1.00) ESR2ESR1KDM4EALDH1A1GAA
SCHEMBL6825266 0.65 ESR2 (1.00) ESR2ESR1KDM4EALDH1A1GAA
SCHEMBL7824164 0.65 KDM4E (0.66) ESR2ESR1KDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894805-B1 Ribose substituted aromatic derivatives, their preparation and use as medicaments AVENTIS PHARMA SA (FR) 2005-02-09 EP disclosed
US-5968939-A ANTIBIOTICS FROM AMINOOXOBENZOPYRAN COMPOUNDS HOECHST MARION ROUSSEL (FR) 1999-10-19 US disclosed
EP-0894805-A1 Ribose substituted aromatic derivatives, their preparation and use as medicaments HOECHST MARION ROUSSEL (FR) 1999-02-03 EP disclosed