SCHEMBL28065504

SCHEMBL28065504

Cc1c(Cl)c(=O)oc2c(O)c(O)ccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 7/20 0.56
ESR1 P03372 6/20 0.56
GAA P10253 5/20 0.56
KDM4E B2RXH2 4/20 0.56
MAPT P10636 2/20 0.56
MAPK1 P28482 2/20 0.56
MCL1 Q07820 2/20 0.56
HTT P42858 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
JAK2 O60674 1/20 0.56
POLB P06746 1/20 0.56
PKM P14618 1/20 0.56
MPI P34949 1/20 0.56
BLM P54132 1/20 0.56
PKLR P30613 1/20 0.54
GALNT2 Q10471 1/20 0.54
GALNT1 Q10472 1/20 0.54
GALNT3 Q14435 1/20 0.54
GALNT10 Q86SR1 1/20 0.54
GALNT13 Q8IUC8 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9211529 0.88 KDM4E (0.66) ESR2ESR1GAAKDM4EMAPK1
SCHEMBL31414410 0.86 KDM4E (0.61) ESR2ESR1GAAKDM4EMAPT
SCHEMBL15285080 0.86 KDM4E (0.61) ESR2ESR1GAAKDM4EMAPT
SCHEMBL10789607 0.80 HSD17B3 (0.50) ESR2ESR1GAAKDM4EHTT
SCHEMBL28065536 0.80 KDM4E (0.79) ESR2ESR1GAAKDM4EMAPT
SCHEMBL28065533 0.80 KDM4E (0.56) ESR2ESR1GAAKDM4EMAPT
SCHEMBL6559867 0.79 ESR1 (0.52) ESR2ESR1GAAKDM4EHTT
SCHEMBL19236367 0.79 KDM4E (0.79) ESR2ESR1GAAKDM4EMAPT
SCHEMBL14756048 0.78 KDM4E (0.53) ESR2ESR1GAAKDM4EMAPT
SCHEMBL8745765 0.75 KDM4E (0.65) ESR2ESR1GAAKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105524034-B Preparation, pharmacological action and the application for treating cerebral ischemia of coumarin derivative 北京大学 2018-08-17 CN disclosed
CN-105566269-B Preparation, pharmacological action and the application for treating itch of coumarin derivative 北京大学 2018-07-10 CN disclosed
CN-105566269-A Preparation and pharmacological effects of coumarin derivative and application of coumarin derivative to treatment on pruritus UNIV BEIJING 2016-05-11 CN disclosed
CN-105524034-A Preparation method of coumarin derivative, pharmacological effect of coumarin derivative and use of coumarin derivative in treatment on cerebral ischemia UNIV BEIJING 2016-04-27 CN disclosed