SCHEMBL6158329

SCHEMBL6158329

CC(C)C(CC(=O)NCCCc1ccccc1)C(=O)NC(CC(=O)O)C(=O)CNS(=O)(=O)CC12CCC(CC1)C2(C)C

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 13/20 0.58
KMT2A Q03164 2/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
CASP3 P42574 2/20 0.35
CASP6 P55212 2/20 0.35
CASP8 Q14790 2/20 0.35
EPHX2 P34913 2/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6160628 0.95 CASP1 (0.61) CASP1CASP3CASP6CASP8
SCHEMBL6158679 0.89 CASP1 (0.74) CASP1KMT2AALDH1A1CYP2C19
SCHEMBL6158315 0.85 CASP1 (0.62) CASP1KMT2AALDH1A1CYP2D6CYP2C9
SCHEMBL6160169 0.84 CASP1 (0.78) CASP1KMT2AALDH1A1CYP2C19
SCHEMBL6157518 0.83 CASP1 (0.69) CASP1KMT2AALDH1A1CYP2C19
SCHEMBL6159134 0.83 CASP1 (0.68) CASP1KMT2AALDH1A1CYP2C19
SCHEMBL6157780 0.82 CASP1 (0.69) CASP1KMT2AALDH1A1CYP2C19
SCHEMBL6159401 0.82 CASP1 (0.67) CASP1KMT2AALDH1A1CYP2C19
SCHEMBL6158325 0.81 CASP1 (0.50) CASP1KMT2AALDH1A1HPGDCASP3
SCHEMBL6159750 0.80 CASP1 (0.75) CASP1KMT2ACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082127-B1 SUCCINAMIDE INHIBITORS OF INTERLEUKIN-1BETA CONVERTING ENZYME WARNER LAMBERT CO (US) 2005-06-22 EP claimed
EP-1082127-B1 SUCCINAMIDE INHIBITORS OF INTERLEUKIN-1BETA CONVERTING ENZYME WARNER LAMBERT CO (US) 2005-06-22 EP disclosed