SCHEMBL6158955

SCHEMBL6158955

CCCNCCC(c1ccccc1)c1cccnc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 4/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
KCNN4 O15554 1/20 0.51
KCNA5 P22460 1/20 0.51
TBXAS1 P24557 1/20 0.49
KCNH2 Q12809 2/20 0.49
CFTR P13569 1/20 0.46
SLC6A2 P23975 1/20 0.46
SLC6A4 P31645 1/20 0.46
SLC6A3 Q01959 1/20 0.46
GOPC Q9HD26 1/20 0.46
HTR2A P28223 1/20 0.46
HRH1 P35367 1/20 0.46
KDM4E B2RXH2 1/20 0.45
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3637324 0.85 KCNH2 (0.63) CYP2C19KCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL23970158 0.84 TBXAS1 (0.56) EPHX2CYP2C9CYP2C19KCNN4KCNA5
SCHEMBL9910965 0.81 TBXAS1 (0.61) EPHX2CYP2C9CYP2C19KCNN4KCNA5
SCHEMBL659775 0.80 CFTR (0.53) EPHX2CYP2C9CYP2C19KCNN4KCNA5
SCHEMBL14288463 0.80 TBXAS1 (0.64) EPHX2CYP2C9CYP2C19KCNN4KCNA5
SCHEMBL15130958 0.77 SLC6A2 (0.70) EPHX2CYP2C9CYP2C19KCNN4KCNA5
SCHEMBL1944201 0.77 CFTR (0.59) KCNN4KCNA5TBXAS1KCNH2CFTR
SCHEMBL11796932 0.76 KCNH2 (0.76) EPHX2CYP2C19KCNH2SLC6A2SLC6A4
SCHEMBL126320 0.75 CASR (0.54) LMNASMN1; SMN2
Ammonia Solution, Strong SCHEMBL5999698 0.75 CFTR (0.57) KCNN4KCNA5TBXAS1KCNH2CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1129070-A4 NEUROTROPHIC DIAMIDE AND CARBAMATE AGENTS BRISTOL MYERS SQUIBB CO (US) 2005-03-02 EP disclosed
EP-1129070-A1 NEUROTROPHIC DIAMIDE AND CARBAMATE AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2001-09-05 EP disclosed
US-6228872-B1 PEPTIDE-PROLYL ISOMERASE AND ROTAMASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY 2001-05-08 US disclosed
WO-2000027811-A1 NEUROTROPHIC DIAMIDE AND CARBAMATE AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2000-05-18 WO disclosed