SCHEMBL6158975

SCHEMBL6158975

O=C1CC(S)CN1Cc1ccc(Oc2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.46
NPBWR1 P48145 1/20 0.41
LTA4H P09960 2/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
HTT P42858 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.39
SIRT1 Q96EB6 1/20 0.39
EGLN1 Q9GZT9 2/20 0.39
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
MMP2 P08253 2/20 0.38
MMP1 P03956 1/20 0.38
MMP3 P08254 1/20 0.38
MMP9 P14780 1/20 0.38
MMP13 P45452 1/20 0.38
MAPK14 Q16539 1/20 0.38
PPARD Q03181 1/20 0.38
PPARA Q07869 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6158458 0.88 GRM2 (0.50) TSHRHCRTR1HCRTR2
SCHEMBL6158131 0.86 HTT (0.54) HPGDTSHRHTTMMP2MMP1
SCHEMBL6158497 0.86 HTT (0.54) HPGDTSHRHTTMMP2MMP1
SCHEMBL6157651 0.84 HPGD (0.54) DPP4HPGDTSHRHRH3HTT
SCHEMBL6158376 0.84 HPGD (0.54) DPP4HPGDTSHRHRH3HTT
SCHEMBL6158698 0.84 HPGD (0.54) DPP4HPGDTSHRHRH3HTT
SCHEMBL6158922 0.84 S1PR5 (0.49) HPGDTSHRHTTEGLN1MMP2
SCHEMBL6158929 0.84 S1PR5 (0.49) HPGDTSHRHTTEGLN1MMP2
SCHEMBL6159859 0.83 PDE4A (0.44) HPGDTSHRHTTMMP2MMP1
SCHEMBL6158478 0.83 HPGD (0.43) HPGDTSHRHTTMMP2MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6953789-B2 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-10-11 US disclosed
US-20040157894-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-08-12 US disclosed
US-6699881-B2 MATRIX METALLOPROTEASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2004-03-02 US disclosed
US-20030078253-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY, LIMITED (JP) 2003-04-24 US disclosed
US-6420415-B1 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
EP-1132379-A1 NOVEL THIOL DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND UTILIZATION THEREOF Takeda Chemical Industries, Ltd. (JP) 2001-09-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030078253-A1 Thiol compounds, their production and use TST, QSOX1, SULT1E1 DPP4 4652/4885NPBWR1 2200/4885LTA4H 1800/4885
US-20040157894-A1 Thiol compounds, their production and use TST, SULT1E1, QSOX1 DPP4 4551/4885NPBWR1 2483/4885LTA4H 1646/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.