SCHEMBL6159448

SCHEMBL6159448

CNc1nc(C)c(-c2ccnc(-c3cc(N)ccc3N)n2)s1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 18/20 0.48
CDK4 P11802 10/20 0.48
CCNA2 P20248 9/20 0.48
PLK1 P53350 1/20 0.48
CDK9 P50750 14/20 0.47
CDK1 P06493 10/20 0.47
CDK7 P50613 10/20 0.47
AURKA O14965 6/20 0.47
AURKB Q96GD4 5/20 0.47
CCNT1 O60563 8/20 0.46
CCNB1 P14635 5/20 0.46
CCNH P51946 5/20 0.46
CCNA1 P78396 3/20 0.46
FLT3 P36888 2/20 0.45
MKNK1 Q9BUB5 1/20 0.45
MKNK2 Q9HBH9 1/20 0.45
CCNE1 P24864 2/20 0.42
WEE1 P30291 2/20 0.41
ALK Q9UM73 2/20 0.41
CHEK1 O14757 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6159471 0.85 CDK2 (0.59) CDK2CDK4PLK1CDK9CDK1
SCHEMBL6409152 0.81 CDK2 (0.65) CDK2CDK4CCNA2CDK9CDK1
SCHEMBL4169064 0.78 CDK2 (0.68) CDK2CDK4CCNA2PLK1CDK9
SCHEMBL7465490 0.78 ALDH1A1 (0.47) CDK2CDK4CDK9CDK1CDK7
SCHEMBL6158084 0.75 CDK2 (0.78) CDK2CDK4CCNA2PLK1CDK9
SCHEMBL5613959 0.72 WEE1 (0.58) CDK2CDK4CCNA2CDK9CDK1
SCHEMBL19554159 0.72 KDM4E (0.41)
SCHEMBL1888365 0.70 CDK2 (0.55) CDK2CDK4CCNA2PLK1CDK9
SCHEMBL29941155 0.69 CDK2 (0.53) CDK2CDK4CCNA2PLK1CDK9
SCHEMBL27624138 0.69 CDK2 (0.61) CDK2CDK4CCNA2PLK1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1581231-A1 ANTI-VIRAL COMPOUNDS Cyclacel Limited (GB) 2005-10-05 EP disclosed
EP-1430051-A1 N-(4-(4-METHYLTHIAZOL-5-YL)PYRIMIDIN-2-YL)-N-PHENYLAMINES AS ANTIPROLIFERATIVE COMPOUNDS Cyclacel Limited (GB) 2004-06-23 EP disclosed
WO-2004043467-A1 ANTI-VIRAL COMPOUNDS CYCLACEL LIMITED (GB) 2004-05-27 WO disclosed
WO-2003029248-A1 N-(4-(4-METHYLTHIAZOL-5-YL) PYRIMIDIN-2-YL) -N-PHENYLAMINES AS ANTIPROLIFERATIVE COMPOUNDS CYCLACEL LIMITED (GB) 2003-04-10 WO disclosed