SCHEMBL7465490

SCHEMBL7465490

Cc1ccsc1-c1ccnc(-c2cc(N)ccc2N)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
HPGD P15428 1/20 0.47
CYP2A6 P11509 7/20 0.42
CYP3A4 P08684 4/20 0.36
CYP2C19 P33261 4/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP1A2 P05177 2/20 0.36
RECQL P46063 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HTT P42858 1/20 0.36
CDK4 P11802 3/20 0.34
CDK2 P24941 3/20 0.34
CCNE1 P24864 1/20 0.34
AURKA O14965 1/20 0.33
CDK1 P06493 1/20 0.33
CDK7 P50613 1/20 0.33
CDK9 P50750 1/20 0.33
HSP90AA1 P07900 1/20 0.33
CYP2B6 P20813 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6159471 0.79 CDK2 (0.59) HTTCDK4CDK2CCNE1AURKA
SCHEMBL7800860 0.78 CYP2A6 (0.50) ALDH1A1CYP2A6CYP3A4CYP2C19CYP2D6
SCHEMBL6159448 0.78 CDK2 (0.48) CDK4CDK2CCNE1AURKACDK1
Hydrochloric Acid SCHEMBL7807397 0.77 CYP2A6 (0.49) ALDH1A1CYP2A6CYP3A4CYP2C19CYP2D6
SCHEMBL7468872 0.76 KDM4E (0.57) ALDH1A1HPGDCYP3A4CYP2C19CYP2D6
SCHEMBL19554159 0.75 KDM4E (0.41) ALDH1A1CYP3A4CYP2C19CYP2C9CYP1A2
SCHEMBL7467076 0.73 KCNH2 (0.41) CYP2A6CDK2CDK9
SCHEMBL7470843 0.72 ALDH1A1 (0.38) ALDH1A1HPGDKDM4EHTTTSHR
SCHEMBL18866730 0.72 ALDH1A1 (0.60) ALDH1A1HPGDCYP2A6CYP3A4CYP2C19
SCHEMBL7476653 0.72 ABL1 (0.48) ALDH1A1CYP3A4CYP2C19CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233461-B2 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 2002-05-29 EP disclosed