SCHEMBL6160249

SCHEMBL6160249

NC(=O)[C@@H]1[C@@H](S)CC(=O)N1Cc1ccc(Oc2ccccc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 3/20 0.44
HCRTR2 O43614 3/20 0.44
HRH3 Q9Y5N1 1/20 0.42
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
FAAH O00519 2/20 0.40
HTT P42858 1/20 0.39
SRD5A2 P31213 2/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
FFAR1 O14842 1/20 0.39
MMP1 P03956 2/20 0.39
MMP2 P08253 2/20 0.39
MMP3 P08254 2/20 0.39
MMP9 P14780 2/20 0.39
MMP13 P45452 2/20 0.39
MMP14 P50281 2/20 0.39
LTA4H P09960 1/20 0.39
PARP10 Q53GL7 1/20 0.38
S1PR5 Q9H228 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6160246 1.00 HCRTR1 (0.44) HCRTR1HCRTR2HRH3NPC1RAB9A
SCHEMBL6160252 1.00 HCRTR1 (0.44) HCRTR1HCRTR2HRH3NPC1RAB9A
SCHEMBL6158494 0.82 HCRTR1 (0.42) HCRTR1HCRTR2HRH3FAAHLTA4H
SCHEMBL6158489 0.82 HCRTR1 (0.42) HCRTR1HCRTR2HRH3FAAHLTA4H
SCHEMBL6158495 0.82 HCRTR1 (0.42) HCRTR1HCRTR2HRH3FAAHLTA4H
SCHEMBL6157435 0.81 HCRTR1 (0.43) HCRTR1HCRTR2HRH3FAAHHTT
SCHEMBL6157425 0.81 HCRTR1 (0.43) HCRTR1HCRTR2HRH3FAAHHTT
SCHEMBL6158372 0.81 HCRTR1 (0.43) HCRTR1HCRTR2HRH3FAAHHTT
SCHEMBL6157986 0.80 HCRTR1 (0.50) HCRTR1HCRTR2HRH3FAAH
SCHEMBL6159559 0.80 HCRTR1 (0.50) HCRTR1HCRTR2HRH3FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6953789-B2 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-10-11 US disclosed
US-20040157894-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-08-12 US disclosed
US-6699881-B2 MATRIX METALLOPROTEASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2004-03-02 US disclosed
US-20030078253-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY, LIMITED (JP) 2003-04-24 US disclosed
US-6420415-B1 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
EP-1132379-A1 NOVEL THIOL DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND UTILIZATION THEREOF Takeda Chemical Industries, Ltd. (JP) 2001-09-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030078253-A1 Thiol compounds, their production and use TST, QSOX1, SULT1E1 HCRTR1 1949/4885HCRTR2 1842/4885HRH3 505/4885
US-20040157894-A1 Thiol compounds, their production and use TST, SULT1E1, QSOX1 HCRTR1 1930/4885HCRTR2 1754/4885HRH3 463/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.