SCHEMBL6160470

SCHEMBL6160470

CC(=O)SCC(Cc1ccccc1F)C(=O)O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CPB2 Q96IY4 1/20 0.43
PPARA Q07869 2/20 0.43
PPARG P37231 1/20 0.43
MME P08473 2/20 0.41
ACE P12821 1/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
ABCC3 O15438 1/20 0.41
NR1I2 O75469 1/20 0.41
ABCB11 O95342 1/20 0.41
NR3C1 P04150 1/20 0.41
RARG P13631 1/20 0.41
CNR1 P21554 1/20 0.41
OPRK1 P41145 1/20 0.41
NR1H2 P55055 1/20 0.41
NR1H3 Q13133 1/20 0.41
NR1I3 Q14994 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7367328 0.84 PPARG (0.45) CPB2PPARAPPARGMMEACE
SCHEMBL7367331 0.84 PPARG (0.45) CPB2PPARAPPARGMMEACE
SCHEMBL7274320 0.82 CYP1A2 (0.55) CPB2PPARAPPARGCYP1A2HPGD
SCHEMBL7318719 0.80 CTNNB1 (0.50) MMEACECYP1A2CYP2C19
SCHEMBL838962 0.80 CYP1A2 (0.63) CPB2PPARAMMECYP1A2CYP3A4
SCHEMBL838961 0.80 CYP1A2 (0.63) CPB2PPARAMMECYP1A2CYP3A4
SCHEMBL14885334 0.80 PPARG (0.49) PPARAPPARGCYP1A2KDM4EALDH1A1
SCHEMBL6154521 0.80 CYP1A2 (0.63) CPB2PPARAMMECYP1A2CYP3A4
Hydrochloric Acid SCHEMBL6572923 0.78 CYP1A2 (0.61) CPB2PPARAMMECYP1A2CYP3A4
Hydrochloric Acid SCHEMBL6572922 0.78 CYP1A2 (0.61) CPB2PPARAMMECYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0877740-B1 THIOL DERIVATIVES WITH METALLOPEPTIDASE INHIBITORY ACTIVITY ZAMBON SPA (IT) 2005-03-30 EP disclosed
US-5994539-A Mercapto acyl aminoacid derivatives endowed with dual ACE-NEP inhibitory activity, useful in the treatment of cardiovascular diseases ZAMBON GROUP S.P.A. (IT) 1999-11-30 US disclosed
US-5760241-A ANGIOTENSIN CONVERTING ENZYME AND ENKEPHALINASE INHIBITORS; CARDIOVASCULAR DISORDERS ZAMBON GROUP S.P.A. (IT) 1998-06-02 US disclosed