SCHEMBL6160581

SCHEMBL6160581

CS(=O)(=O)OC1c2ccccc2CSc2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
GAA P10253 2/20 0.49
MAPT P10636 5/20 0.47
HPGD P15428 2/20 0.47
ALOX12 P18054 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
POLB P06746 1/20 0.41
TBXA2R P21731 1/20 0.37
KMT2A Q03164 3/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B3 P37058 1/20 0.35
MEN1 O00255 2/20 0.35
RAD52 P43351 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
USP2 O75604 1/20 0.34
LMNA P02545 1/20 0.33
THRB P10828 1/20 0.33
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22891090 0.79 ABCB11 (0.38) ALDH1A1GAAUSP2
SCHEMBL23386681 0.79 ABCB11 (0.38) ALDH1A1GAAUSP2
SCHEMBL14997683 0.75 ALDH1A1 (0.55) ALDH1A1GAAMAPTHPGDALOX12
SCHEMBL19718931 0.74 ALDH1A1 (0.54) ALDH1A1GAAMAPTHPGDALOX12
SCHEMBL5466833 0.73 ALDH1A1 (0.57) ALDH1A1GAAMAPTHPGDALOX12
SCHEMBL9610482 0.72 ALDH1A1 (0.52) ALDH1A1GAAMAPTHPGDALOX12
Sevitropium SCHEMBL1816494 0.72 CHRNA7 (0.44) ALDH1A1GAAMAPTHPGDALOX12
SCHEMBL21185020 0.72 ALDH1A1 (0.55) ALDH1A1GAAMAPTHPGDALOX12
SCHEMBL10239427 0.72 ALDH1A1 (0.55) ALDH1A1GAAMAPTHPGDALOX12
SCHEMBL3846181 0.71 CA1 (0.42) ALDH1A1MAPTHPGDTDP1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1060163-B1 NEW PIPERAZINYL-SUBSTITUTED PYRIDYLALKANE, ALKENE AND ALKINE CARBOXAMIDES KLINGE CO CHEM PHARM FAB (DE) 2005-10-12 EP disclosed
US-6903118-B1 Piperazinyl-substituted pyridylalkane, alkene and alkine carboxamides KLINGE PHARMA GMBH (DE) 2005-06-07 US disclosed