SCHEMBL6160979

SCHEMBL6160979

CCCc1nc(Sc2ccc(CC(=O)O)cc2)c(C(=O)O)n1Cc1cc2c(cc1Cl)OCO2

nearest known ligand 0.63

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 4/20 0.63
AGTR1 P30556 4/20 0.45
AGTR2 P50052 4/20 0.45
SLC22A12 Q96S37 1/20 0.45
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
EDNRB P24530 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6159406 0.91 EDNRA (0.63) EDNRAAGTR1AGTR2KDM4EALDH1A1
SCHEMBL8434286 0.90 EDNRA (0.64) EDNRAAGTR1AGTR2KDM4EALDH1A1
SCHEMBL6162876 0.88 EDNRA (0.60) EDNRAAGTR1AGTR2KDM4EALDH1A1
SCHEMBL7498870 0.85 EDNRA (0.59) EDNRAAGTR1AGTR2KDM4EALDH1A1
SCHEMBL3837125 0.84 EDNRA (0.70) EDNRAAGTR1AGTR2KDM4EALDH1A1
SCHEMBL7501757 0.83 EDNRA (0.55) EDNRAEDNRB
SCHEMBL8431316 0.82 EDNRA (0.52) EDNRASLC22A12KDM4EALDH1A1HPGD
SCHEMBL8434768 0.81 EDNRA (0.52) EDNRAKDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL7496869 0.80 EDNRA (0.66) EDNRAAGTR1AGTR2SLC22A12KDM4E
SCHEMBL7502689 0.79 EDNRA (0.54) EDNRAAGTR1AGTR2SLC22A12KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863896-B1 NOVEL IMIDAZOLE DERIVATIVES, METHOD FOR PREPARING SAME, PHARMACEUTICAL COMPOSITIONS AND USE OF SAID DERIVATIVES AS ENDOTHELIN ANTAGONISTS AVENTIS PHARMA SA (FR) 2005-02-09 EP claimed