SCHEMBL8434286

SCHEMBL8434286

CCCc1nc(Sc2ccc3c(c2)OCO3)c(C(=O)O)n1Cc1cc2c(cc1Cl)OCO2

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 9/20 0.64
AGTR1 P30556 1/20 0.46
AGTR2 P50052 1/20 0.46
EDNRB P24530 8/20 0.44
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ITGB2 P05107 1/20 0.37
ICAM1 P05362 1/20 0.37
ITGAL P20701 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6159406 0.92 EDNRA (0.63) EDNRAAGTR1AGTR2KDM4EALDH1A1
SCHEMBL7498870 0.90 EDNRA (0.59) EDNRAAGTR1AGTR2EDNRBKDM4E
SCHEMBL6160979 0.90 EDNRA (0.63) EDNRAAGTR1AGTR2EDNRBKDM4E
SCHEMBL6162876 0.87 EDNRA (0.60) EDNRAAGTR1AGTR2EDNRBKDM4E
SCHEMBL3837125 0.87 EDNRA (0.70) EDNRAAGTR1AGTR2KDM4EALDH1A1
SCHEMBL7501757 0.85 EDNRA (0.55) EDNRAEDNRB
SCHEMBL8434768 0.82 EDNRA (0.52) EDNRAEDNRBKDM4EALDH1A1HPGD
SCHEMBL7498348 0.81 EDNRA (0.63) EDNRAAGTR1AGTR2KDM4EALDH1A1
SCHEMBL8434967 0.81 EDNRA (0.63) EDNRAAGTR1AGTR2
SCHEMBL7496869 0.81 EDNRA (0.66) EDNRAAGTR1AGTR2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5932741-A TREATING ILLNESSES RESULTING FROM ABNORMAL STIMULATION OF ENDOTHELIN RECEPTORS HOECHST MARION ROUSSEL (FR) 1999-08-03 US disclosed
US-5811444-A IMIDAZOLE DERIVATIVES ROUSSEL UCLAF (FR) 1998-09-22 US disclosed