SCHEMBL6161012

SCHEMBL6161012

Cc1ccccc1-c1nc(NC(=O)Nc2cccc(C(=O)OCc3ccccc3)c2)c(CCC23CC4CC(CC(C4)C2)C3)n1C(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PPIA P62937 2/20 0.41
EPHX2 P34913 1/20 0.40
CCKBR P32239 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7087125 0.92 PPIA (0.43) PPIACCKBRRAB9A
SCHEMBL7083915 0.86 NPC1 (0.37) EPHX2RAB9A
SCHEMBL6157991 0.83 EPHX2 (0.35) EPHX2
SCHEMBL6330062 0.82 EPHX2 (0.37) EPHX2
SCHEMBL7677952 0.81
SCHEMBL6160443 0.81 PPIA (0.45) PPIA
SCHEMBL7080456 0.80
SCHEMBL7688902 0.77 RAB9A (0.40) CCKBRRAB9A
SCHEMBL6158866 0.75 P2RX7 (0.34)
SCHEMBL7086457 0.74 P2RX7 (0.35) EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1492784-A2 SUBSTITUTED 2,3-DIPHENYL PYRIDINES Merck & Co., Inc. (US) 2005-01-05 EP disclosed
WO-2003082191-A2 SUBSTITUTED 2,3-DIPHENYL PYRIDINES MERCK & CO., INC. (US) 2003-10-09 WO disclosed
US-6479531-B1 Gastrin and cholecystokinin receptor ligands JAMES BLACK FOUNDATION LIMITED (GB) 2002-11-12 US disclosed