SCHEMBL6161584

SCHEMBL6161584

COc1ccc(C(=O)CCc2ccc(NC3=NCCN3)cc2)c(F)c1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGIR P43119 13/20 0.58
ADRA2A P08913 5/20 0.56
ADRA2B P18089 4/20 0.56
ADRA2C P18825 4/20 0.56
GPR65 Q8IYL9 1/20 0.47
WDR5 P61964 1/20 0.47
AOC3 Q16853 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6161381 0.99 PTGIR (0.57) PTGIRADRA2AADRA2BADRA2CGPR65
SCHEMBL6159356 0.88 ADRA2A (0.50) PTGIRADRA2AADRA2BADRA2CGPR65
Hydrochloric Acid SCHEMBL6161371 0.87 ADRA2A (0.49) PTGIRADRA2AADRA2BADRA2CGPR65
SCHEMBL5658067 0.85 WDR5 (0.60) PTGIRADRA2AADRA2BADRA2CGPR65
SCHEMBL6160627 0.83 ADRA2A (0.52) PTGIRADRA2AADRA2BADRA2CGPR65
SCHEMBL6158402 0.83 PTGIR (0.63) PTGIRADRA2AADRA2BADRA2CGPR65
Hydrochloric Acid SCHEMBL6161625 0.81 ADRA2A (0.49) PTGIRADRA2AADRA2BADRA2CWDR5
SCHEMBL6159168 0.80 ADRA2A (0.48) PTGIRADRA2AADRA2BADRA2CGPR65
SCHEMBL6159740 0.80 ADRA2A (0.50) PTGIRADRA2AADRA2BADRA2CAOC3
SCHEMBL6056621 0.79 ADRA2A (0.45) PTGIRADRA2AADRA2BADRA2CAOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339694-B1 SUBSTITUTED 2-PHENYLAMINOIMIDAZOLINE PHENYL KETONE DERIVATIVES AS IP ANTAGONISTS HOFFMANN LA ROCHE (CH) 2005-09-21 EP disclosed
EP-1339694-A1 SUBSTITUTED 2-PHENYLAMINOIMIDAZOLINE PHENYL KETONE DERIVATIVES AS IP ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2003-09-03 EP disclosed
US-6417186-B1 TREATING PAIN, URINARY TRACT INFECTIONS, INFLAMMATION, RESPIRATORY DISEASE STATES FROM ALLERGIES OR ASTHMA, EDEMA FORMATION OR HYPOTENSIVE VASCULAR DISEASES. SYNTEX (U.S.A.) LLC 2002-07-09 US disclosed
WO-2002040453-A1 SUBSTITUTED 2-PHENYLAMINOIMIDAZOLINE PHENYL KETONE DERIVATIVES AS IP ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2002-05-23 WO disclosed