SCHEMBL6162009

SCHEMBL6162009

COC(=O)c1cc([N+](=O)[O-])ccc1NC(=O)OC(C)(C)C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.53
HTT P42858 1/20 0.53
ALOX5 P09917 1/20 0.48
POLB P06746 1/20 0.48
ALDH1A1 P00352 4/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 5/20 0.47
GLA P06280 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CTSV O60911 1/20 0.44
CTSL P07711 1/20 0.44
NR3C2 P08235 1/20 0.44
MMP1 P03956 1/20 0.43
MMP2 P08253 1/20 0.43
MMP9 P14780 1/20 0.43
MMP8 P22894 1/20 0.43
MMP13 P45452 1/20 0.43
ATR Q13535 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7594732 0.90 SMN1; SMN2 (0.54) PKMHTTALOX5POLBALDH1A1
SCHEMBL1082203 0.88 MEN1 (0.49) PKMHTTALOX5POLBALDH1A1
SCHEMBL9307475 0.88 SMN1; SMN2 (0.59) PKMHTTALOX5POLBALDH1A1
SCHEMBL17085330 0.88 PKM (0.68) PKMHTTPOLBALDH1A1GAA
SCHEMBL5285260 0.83 PKM (0.78) PKMHTTPOLBALDH1A1GAA
SCHEMBL1954190 0.83 CXCR1 (0.54) PKMHTTALOX5POLBALDH1A1
SCHEMBL28573397 0.83 NPC1 (0.60) PKMHTTPOLBALDH1A1MAPT
SCHEMBL15160073 0.83 HTT (0.53) PKMHTTALOX5POLBALDH1A1
SCHEMBL5629195 0.82 SMN1; SMN2 (0.60) PKMHTTPOLBALDH1A1GAA
SCHEMBL2831541 0.82 MAPT (0.53) PKMHTTALOX5POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1178969-B1 GASTRIN AND CHOLECYSTOKININ RECEPTOR LIGANDS BLACK JAMES FOUNDATION (GB) 2005-07-13 EP disclosed
EP-0593603-B1 BICYCLIC FIBRINOGEN ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2002-11-20 EP disclosed
US-6479531-B1 Gastrin and cholecystokinin receptor ligands JAMES BLACK FOUNDATION LIMITED (GB) 2002-11-12 US disclosed
EP-1178969-A1 GASTRIN AND CHOLECYSTOKININ RECEPTOR LIGANDS JAMES BLACK FOUNDATION LIMITED (GB) 2002-02-13 EP disclosed
US-6127359-A Bicyclic fibrinogen antagonists SMITHKLINE BEECHAM CORPORATION (US) 2000-10-03 US disclosed
WO-2000027823-A1 GASTRIN AND CHOLECYSTOKININ RECEPTOR LIGANDS JAMES BLACK FOUNDATION LIMITED (GB) 2000-05-18 WO disclosed
US-5939412-A Bicyclic fibrinogen antagonists SMITHKLINE BEECHAM CORPORATION (US) 1999-08-17 US disclosed
US-5693636-A Bicyclic fibrinogen antagonists SMITHKLINE BEECHAM CORPORATION (US) 1997-12-02 US disclosed
EP-0593603-A1 BICYCLIC FIBRINOGEN ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1994-04-27 EP disclosed
WO-1993000095-A2 BICYCLIC FIBRINOGEN ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1993-01-07 WO disclosed