SCHEMBL6162544

SCHEMBL6162544

O=C=NC(=O)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TPMT P51580 1/20 0.48
HCAR1 Q9BXC0 1/20 0.38
RXRA P19793 2/20 0.35
RXRB P28702 2/20 0.35
RAB9A P51151 1/20 0.35
TSHR P16473 1/20 0.35
FLT1 P17948 1/20 0.33
FLT4 P35916 1/20 0.33
KDR P35968 1/20 0.33
FABP4 P15090 1/20 0.33
ATM Q13315 1/20 0.33
HCAR2 Q8TDS4 1/20 0.32
PARP1 P09874 1/20 0.32
TTR P02766 1/20 0.32
HTR3E A5X5Y0 1/20 0.31
HTR3B O95264 1/20 0.31
HTR3A P46098 1/20 0.31
HTR3D Q70Z44 1/20 0.31
HTR3C Q8WXA8 1/20 0.31
GRN P28799 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1789230 0.84
SCHEMBL5825164 0.81 TPMT (0.46) TPMTHCAR1RXRARXRBRAB9A
SCHEMBL10792089 0.80 PARP1 (0.53) RAB9AFLT1FLT4KDRPARP1
SCHEMBL9381338 0.79 S1PR2 (0.39)
SCHEMBL3205731 0.78 CES2 (0.50) RAB9ATSHR
SCHEMBL6282074 0.76 TPMT (0.42) TPMTHCAR1RXRARXRBRAB9A
SCHEMBL3208606 0.74 TPMT (0.48) TPMTHCAR1RXRARXRBRAB9A
SCHEMBL3393415 0.74 TP53 (0.36) TSHR
SCHEMBL10999100 0.74 TSHR (0.53) RAB9ATSHR
SCHEMBL12534325 0.73 TPMT (0.52) TPMTHCAR1RXRARXRBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0893442-B1 LYMPH-ABSORBABLE IMIDAZOLE DERIVATIVES SHIONOGI & CO (JP) 2005-01-12 EP disclosed
US-6054591-A LYMPHOTROPIC ANTI-AIDS AGENT SHIONOGI & CO., LTD. (JP) 2000-04-25 US disclosed
EP-0893442-A1 LYMPH-ABSORBABLE IMIDAZOLE DERIVATIVES SHIONOGI & CO., LTD. (JP) 1999-01-27 EP disclosed
US-5106843-A Treatment of migraine, emesis, anxiety, gastrointestinal disorders, psychological disorders AMERICAN HOME PRODUCTS CORPORATION (US) 1992-04-21 US disclosed
EP-0323077-B1 HETEROCYCLIC COMPOUNDS JOHN WYETH & BROTHER LIMITED (GB) 1991-09-11 EP disclosed
US-4983600-A Antiemetics, antianxiety agents, gastrointestinal disorders JOHN WYETH & BROTHER LIMITED (GB) 1991-01-08 US disclosed
EP-0323077-A1 Heterocyclic compounds JOHN WYETH & BROTHER LIMITED (GB) 1989-07-05 EP disclosed
US-4698333-A Use of substituted malonic acid derivatives as agents for combating pests BAYER AKTIENGESELLSCHAFT (DE) 1987-10-06 US disclosed
US-4150158-A Oxadiazindione derivatives useful as insecticides IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1979-04-17 US disclosed