SCHEMBL6163570

SCHEMBL6163570

CN(C)C1(c2ccccc2)CCC(CNC(=O)CCCCCc2c[nH]c3ccc(F)cc23)CC1

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 6/20 0.61
OPRM1 P35372 5/20 0.61
MPO P05164 5/20 0.54
TRPV1 Q8NER1 3/20 0.45
SLC6A4 P31645 3/20 0.45
MTNR1A P48039 3/20 0.43
MTNR1B P49286 3/20 0.43
NOTUM Q6P988 1/20 0.43
SPR P35270 1/20 0.42
HTR1A P08908 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6159000 0.99 OPRL1 (0.62) OPRL1OPRM1MPOTRPV1SLC6A4
SCHEMBL6161294 0.97 OPRL1 (0.63) OPRL1OPRM1MPOSLC6A4MTNR1A
SCHEMBL6160062 0.90 OPRL1 (0.49) OPRL1OPRM1TRPV1SLC6A4MTNR1A
SCHEMBL6165082 0.90 OPRL1 (0.58) OPRL1OPRM1MTNR1A
SCHEMBL6168849 0.89 OPRL1 (0.59) OPRL1OPRM1MTNR1A
SCHEMBL4851081 0.86 OPRL1 (0.69) OPRL1OPRM1MPOMTNR1AMTNR1B
Hydrochloric Acid SCHEMBL5339275 0.86 OPRL1 (0.60) OPRL1OPRM1MTNR1A
Citric Acid SCHEMBL4849030 0.80 OPRL1 (0.60) OPRL1OPRM1TRPV1MTNR1AMTNR1B
SCHEMBL4850795 0.78 OPRL1 (0.76) OPRL1OPRM1MPOMTNR1AMTNR1B
SCHEMBL5234590 0.78 OPRL1 (0.60) OPRL1OPRM1MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562891-A1 4-AMINOMETHYL-1-ARYL-CYCLOHEXYLAMINE DERIVATIVES Grünenthal GmbH (DE) 2005-08-17 EP claimed
WO-2004043899-A1 4-AMINOMETHYL-1-ARYL-CYCLOHEXYLAMINE DERIVATIVES Grünenthal GmbH (DE) 2004-05-27 WO claimed
EP-1562891-A1 4-AMINOMETHYL-1-ARYL-CYCLOHEXYLAMINE DERIVATIVES Grünenthal GmbH (DE) 2005-08-17 EP disclosed
WO-2004043899-A1 4-AMINOMETHYL-1-ARYL-CYCLOHEXYLAMINE DERIVATIVES Grünenthal GmbH (DE) 2004-05-27 WO disclosed