SCHEMBL6164099

SCHEMBL6164099

CCCc1nn(CCO)c2c1C(=O)CCC2

nearest known ligand 0.66

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.66
ALPL P05186 1/20 0.40
ALDH1A1 P00352 3/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
LMNA P02545 2/20 0.34
TSHR P16473 1/20 0.34
PLK1 P53350 1/20 0.32
CSNK2A1 P68400 1/20 0.32
PLK3 Q9H4B4 1/20 0.32
BUB1 O43683 2/20 0.31
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6166704 0.82 HTT (0.64) HTTLMNATSHRPLK1CSNK2A1
SCHEMBL6165467 0.81 ALDH1A1 (0.45) HTTALPLALDH1A1MAPTKMT2A
SCHEMBL6165167 0.80 HTT (1.00) HTTALDH1A1LMNATSHRPLK1
SCHEMBL6163497 0.78 HTT (0.40) HTTALPLALDH1A1KMT2ANPSR1
SCHEMBL6167101 0.76 HTT (0.56) HTT
SCHEMBL6164656 0.76 HTT (0.68) HTTPLK1CSNK2A1PLK3BUB1
SCHEMBL6165245 0.76 HTT (0.68) HTTALDH1A1NPSR1LMNATSHR
SCHEMBL6164449 0.76 HTT (0.38) HTTALPLALDH1A1KMT2ANPSR1
SCHEMBL6167721 0.75 HTT (0.48) HTT
SCHEMBL6168258 0.74 HTT (0.65) HTTPLK1CSNK2A1PLK3BUB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-B1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-04-20 EP disclosed
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed