SCHEMBL6165418

SCHEMBL6165418

CCOC(=O)/C=C/c1ccc(Nc2ncnc3cc(OCc4ccccc4)c(OC)cc23)cc1

nearest known ligand 0.68

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EGFR P00533 10/20 0.68
KDR P35968 9/20 0.60
ABCG2 Q9UNQ0 3/20 0.58
ERBB2 P04626 1/20 0.57
ERBB4 Q15303 1/20 0.57
HDAC3 O15379 1/20 0.57
HDAC1 Q13547 1/20 0.57
HDAC6 Q9UBN7 1/20 0.57
AURKB Q96GD4 2/20 0.55
AURKA O14965 1/20 0.55
RET P07949 1/20 0.55
ABCB1 P08183 2/20 0.55
LCK P06239 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6162952 0.92 KDR (0.70) EGFRKDRABCG2HDAC3HDAC1
SCHEMBL6162829 0.92 KDR (0.70) EGFRKDRABCG2HDAC3HDAC1
SCHEMBL6165325 0.90 EGFR (0.73) EGFRKDRABCG2ERBB2ERBB4
SCHEMBL6165317 0.90 EGFR (0.73) EGFRKDRABCG2ERBB2ERBB4
SCHEMBL6164322 0.81 ABCG2 (0.73) EGFRKDRABCG2HDAC3HDAC1
SCHEMBL6162864 0.81 ABCG2 (0.73) EGFRKDRABCG2HDAC3HDAC1
SCHEMBL3529976 0.81 ABCG2 (0.73) EGFRKDRABCG2HDAC3HDAC1
SCHEMBL30891782 0.81 EGFR (0.83) EGFRKDRERBB2RETLCK
SCHEMBL6686765 0.81 EGFR (0.79) EGFRKDRERBB2ERBB4AURKB
SCHEMBL6164038 0.81 HDAC1 (0.71) EGFRKDRABCG2ERBB2ERBB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218357-B1 QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2005-04-06 EP claimed