SCHEMBL6165317

SCHEMBL6165317

COc1cc2c(Nc3ccc(/C=C/C(=O)O)cc3)ncnc2cc1OCc1ccccc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 10/20 0.73
ABCG2 Q9UNQ0 4/20 0.62
KDR P35968 4/20 0.62
HDAC3 O15379 1/20 0.61
HDAC1 Q13547 1/20 0.61
HDAC6 Q9UBN7 1/20 0.61
RET P07949 2/20 0.60
AURKB Q96GD4 4/20 0.60
AURKA O14965 1/20 0.60
ERBB2 P04626 1/20 0.59
ERBB4 Q15303 1/20 0.59
LCK P06239 2/20 0.59
ABCB1 P08183 3/20 0.59
IRAK4 Q9NWZ3 2/20 0.58
RIPK2 O43353 2/20 0.58
GAK O14976 1/20 0.58
STK10 O94804 1/20 0.58
FLT3 P36888 1/20 0.58
JAK3 P52333 1/20 0.58
AAK1 Q2M2I8 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6165325 1.00 EGFR (0.73) EGFRABCG2KDRHDAC3HDAC1
SCHEMBL3529976 0.91 ABCG2 (0.73) EGFRABCG2KDRHDAC3HDAC1
SCHEMBL6164322 0.91 ABCG2 (0.73) EGFRABCG2KDRHDAC3HDAC1
SCHEMBL6162864 0.91 ABCG2 (0.73) EGFRABCG2KDRHDAC3HDAC1
SCHEMBL6165418 0.90 EGFR (0.68) EGFRABCG2KDRHDAC3HDAC1
SCHEMBL30891782 0.85 EGFR (0.83) EGFRKDRRETERBB2LCK
SCHEMBL6686765 0.85 EGFR (0.79) EGFRKDRRETAURKBAURKA
SCHEMBL6162938 0.84 KDR (0.74) EGFRABCG2KDRHDAC3HDAC1
SCHEMBL6162947 0.84 KDR (0.74) EGFRABCG2KDRHDAC3HDAC1
SCHEMBL6684007 0.84 EGFR (0.74) EGFRKDRRETAURKBAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218357-B1 QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2005-04-06 EP claimed