SCHEMBL6165569

SCHEMBL6165569

O=C(CO)c1cccc(NC(=O)c2ccc(OCCCCc3ccccc3)cc2)c1

nearest known ligand 0.83

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 15/20 0.83
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
CYSLTR1 Q9Y271 2/20 0.54
NPC1 O15118 2/20 0.54
POLB P06746 1/20 0.53
RAB9A P51151 1/20 0.53
SENP8 Q96LD8 1/20 0.53
SENP7 Q9BQF6 1/20 0.53
SENP6 Q9GZR1 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8119505 1.00 NR1H4 (0.83) NR1H4MEN1KMT2ACYSLTR1NPC1
SCHEMBL6577552 0.99 NR1H4 (0.82) NR1H4MEN1KMT2ACYSLTR1NPC1
SCHEMBL8108301 0.97 NR1H4 (0.78) NR1H4MEN1KMT2ANPC1POLB
SCHEMBL6581896 0.93 NR1H4 (0.72) NR1H4MEN1KMT2ANPC1POLB
SCHEMBL6577998 0.90 NR1H4 (0.65) NR1H4MEN1KMT2APOLBRAB9A
SCHEMBL6577802 0.87 NR1H4 (0.62) NR1H4MEN1KMT2APOLBRAB9A
SCHEMBL6577743 0.86 NR1H4 (0.80) NR1H4MEN1KMT2ANPC1POLB
SCHEMBL7476886 0.86 NR1H4 (0.66) NR1H4MEN1KMT2ACYSLTR1NPC1
SCHEMBL6577705 0.85 NR1H4 (0.78) NR1H4MEN1KMT2ANPC1RAB9A
SCHEMBL8827735 0.84 NR1H4 (0.59) NR1H4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111960957-A Preparation method of pranlukast intermediate 太仓康源化建医药有限公司 2020-11-20 CN claimed
CN-108912100-A A kind of preparation method of Pranlukast 浙江三门恒康制药有限公司 2018-11-30 CN claimed
EP-0920427-B1 PROCESS FOR THE PREPARATION OF BENZOPYRAN COMPOUNDS SMITHKLINE BEECHAM PLC (GB) 2002-11-20 EP claimed
US-6048983-A Process for the preparation of benzopyran compounds SMITHKLINE BEECHAM PL.C (GB) 2000-04-11 US claimed
EP-0920427-A1 PROCESS FOR THE PREPARATION OF BENZOPYRAN COMPOUNDS SMITHKLINE BEECHAM PLC (GB) 1999-06-09 EP claimed
WO-1998006718-A1 PROCESS FOR THE PREPARATION OF BENZOPYRAN COMPOUNDS SMITHKLINE BEECHAM PLC (GB) 1998-02-19 WO claimed
JP-9071558-A None JP disclosed
CN-111960957-A Preparation method of pranlukast intermediate 太仓康源化建医药有限公司 2020-11-20 CN disclosed
CN-111960957-A Preparation method of pranlukast intermediate 太仓康源化建医药有限公司 2020-11-20 CN disclosed
CN-108912100-A A kind of preparation method of Pranlukast 浙江三门恒康制药有限公司 2018-11-30 CN disclosed
EP-0964861-B1 PROCESS FOR THE PRODUCTION OF TETRAZOLYLBENZOPYRANS SMITHKLINE BEECHAM PLC (GB) 2005-04-27 EP disclosed
EP-0716088-B1 PROCESS FOR PRODUCING 2-(TETRAZOL-5-YL)-4-OXO-4H-BENZOPYRANS SUMITOMO CHEMICAL CO (JP) 2004-02-18 EP disclosed
EP-0670835-B1 PROCESS FOR PREPARING BENZOPYRAN COMPOUNDS SMITHKLINE BEECHAM PLC (GB) 2003-03-12 EP disclosed
US-5597929-A Production process of 2-(tetrazol-5-yl)-4-oxo-4H-benzopyran SUMITOMO CHEMICAL CO., LTD. (JP) 1997-01-28 US disclosed
US-5596103-A Process for preparing benzopyran compounds SMITHKLINE BEECHAM PLC (GB) 1997-01-21 US disclosed
US-5587483-A Process for preparing tetrazol-5-yl substituted benzopyran compounds SMITHKLINE BEECHAM PLC (GB) 1996-12-24 US disclosed
EP-0716088-A1 PROCESS FOR PRODUCING 2-(TETRAZOL-5-YL)-4-OXO-4H-BENZOPYRANS SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-06-12 EP disclosed
WO-1995032199-A1 PROCESS FOR PREPARING BENZOPYRAN COMPOUNDS SMITHKLINE BEECHAM PLC (GB) 1995-11-30 WO disclosed
EP-0670835-A1 PROCESS FOR PREPARING BENZOPYRAN COMPOUNDS SMITHKLINE BEECHAM PLC (GB) 1995-09-13 EP disclosed
WO-1994012492-A1 PROCESS FOR PREPARING BENZOPYRAN COMPOUNDS SMITHKLINE BEECHAM PLC (GB) 1994-06-09 WO disclosed