SCHEMBL6166997

SCHEMBL6166997

COC(=O)c1ccc(-c2ccc(N)cc2)c(C)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.54
EGFR P00533 1/20 0.49
MAPT P10636 4/20 0.49
KDM4E B2RXH2 4/20 0.49
ALDH1A1 P00352 3/20 0.49
GAA P10253 2/20 0.49
HPGD P15428 2/20 0.49
HSD17B10 Q99714 2/20 0.49
GLA P06280 1/20 0.49
CASP1 P29466 1/20 0.49
CASP7 P55210 1/20 0.49
ATM Q13315 1/20 0.49
PTGS2 P35354 1/20 0.47
HSD17B1 P14061 1/20 0.46
RAB9A P51151 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
TP53 P04637 1/20 0.45
CA12 O43570 2/20 0.45
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6102320 0.91 SLC2A1 (0.58) SLC2A1EGFRMAPTKDM4EALDH1A1
SCHEMBL28255681 0.90 SLC2A1 (0.63) SLC2A1EGFRMAPTKDM4EALDH1A1
SCHEMBL4765793 0.88 MAPT (0.49) SLC2A1EGFRMAPTKDM4EALDH1A1
SCHEMBL6883774 0.86 HSD17B1 (0.59) SLC2A1EGFRMAPTKDM4EALDH1A1
SCHEMBL7402540 0.86 SLC2A1 (0.56) SLC2A1EGFRKDM4EALDH1A1GAA
SCHEMBL8134690 0.85 SLC2A1 (0.52) SLC2A1EGFRMAPTKDM4EALDH1A1
SCHEMBL1528983 0.84 CA1 (0.61) SLC2A1EGFRMAPTKDM4EALDH1A1
SCHEMBL12002526 0.84 SLC2A1 (0.54) SLC2A1EGFRMAPTKDM4EALDH1A1
SCHEMBL4710854 0.84 SLC2A1 (0.54) SLC2A1EGFRMAPTKDM4EALDH1A1
SCHEMBL4465627 0.84 RARB (0.51) SLC2A1EGFRALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1368337-B1 PIPERAZINE DERIVATIVES AND THEIR USE AS 5-HT1B LIGANDS SMITHKLINE BEECHAM PLC (GB) 2005-06-15 EP disclosed