SCHEMBL6167224

SCHEMBL6167224

Cc1nc2ccncc2n1C1C[C@H]2CC[C@@H](C1)N2C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 15/20 0.42
KCNH2 Q12809 3/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
LMNA P02545 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP11B2 P19099 1/20 0.38
AOC3 Q16853 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
OGFRL1 Q5TC84 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6167230 1.00 CCR5 (0.42) CCR5KCNH2L3MBTL1LMNACYP2D6
SCHEMBL4011542 0.90 CCR5 (0.42) CCR5KCNH2L3MBTL1LMNACYP2D6
SCHEMBL4011538 0.90 CCR5 (0.42) CCR5KCNH2L3MBTL1LMNACYP2D6
SCHEMBL3064218 0.81 CCR5 (0.47) CCR5KCNH2L3MBTL1LMNACYP2D6
SCHEMBL3064217 0.81 CCR5 (0.47) CCR5KCNH2L3MBTL1LMNACYP2D6
SCHEMBL13834246 0.77 CCR5 (0.40) CCR5L3MBTL1LMNACYP2D6CYP11B2
SCHEMBL13834245 0.77 CCR5 (0.40) CCR5L3MBTL1LMNACYP2D6CYP11B2
SCHEMBL4134072 0.77 DYRK1A (0.53) CCR5L3MBTL1LMNACYP2D6
SCHEMBL4901353 0.77 CYP11B2 (0.38) CCR5KCNH2CYP2D6CYP11B2AOC3
SCHEMBL4902112 0.77 CYP11B2 (0.40) CCR5KCNH2LMNACYP11B2AOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569646-A2 PIPERIDINE DERIVATIVES AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2005-09-07 EP disclosed
WO-2004054974-A2 PIPERIDINE DERIVATIVES AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2004-07-01 WO disclosed