SCHEMBL6167737

SCHEMBL6167737

Cc1ccc(CNC(=O)c2cccnc2)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.74
NAMPT P43490 4/20 0.72
MMP13 P45452 1/20 0.64
ALDH1A1 P00352 1/20 0.63
HDAC3 O15379 1/20 0.63
HDAC4 P56524 1/20 0.63
HDAC1 Q13547 1/20 0.63
HDAC7 Q8WUI4 1/20 0.63
HDAC2 Q92769 1/20 0.63
HDAC10 Q969S8 1/20 0.63
HDAC11 Q96DB2 1/20 0.63
HDAC8 Q9BY41 1/20 0.63
HDAC6 Q9UBN7 1/20 0.63
HDAC9 Q9UKV0 1/20 0.63
HDAC5 Q9UQL6 1/20 0.63
SMN1; SMN2 Q16637 2/20 0.62
HPGD P15428 2/20 0.62
LMNA P02545 1/20 0.62
GLA P06280 1/20 0.62
POLB P06746 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8372128 0.88 TSHR (0.74) TSHRNAMPTALDH1A1HDAC3HDAC4
SCHEMBL19358859 0.88 ALDH1A1 (0.84) TSHRNAMPTALDH1A1SMN1; SMN2LMNA
SCHEMBL3918322 0.87 TSHR (0.76) TSHRNAMPTALDH1A1HDAC3HDAC4
SCHEMBL354041 0.86 TSHR (0.76) TSHRNAMPTHDAC3HDAC4HDAC1
SCHEMBL19028142 0.86 TSHR (0.76) TSHRNAMPTMMP13HDAC3HDAC4
SCHEMBL5078944 0.86 TSHR (0.71) TSHRNAMPTMMP13ALDH1A1HDAC3
SCHEMBL13102334 0.85 MMP13 (0.85) TSHRNAMPTMMP13ALDH1A1SMN1; SMN2
SCHEMBL29437161 0.85 MMP13 (0.85) TSHRNAMPTMMP13ALDH1A1SMN1; SMN2
SCHEMBL28793879 0.85 TSHR (0.74) TSHRNAMPTHDAC3HDAC4HDAC1
Iodide SCHEMBL15903217 0.85 TSHR (0.74) TSHRNAMPTHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537085-A1 OXYTOCIN INHIBITORS Pfizer Limited (GB) 2005-06-08 EP claimed
WO-2004020414-A1 OXYTOCIN INHIBITORS PFIZER LIMITED (GB) 2004-03-11 WO claimed
EP-2443123-B1 SMALL MOLECULE INHIBITORS OF SPLEEN TYROSINE KINASE (SYK) RIGEL PHARMACEUTICALS INC (US) 2017-04-05 EP disclosed