SCHEMBL6168326

SCHEMBL6168326

CCNc1ncccc1C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 5/20 0.58
ALDH1A1 P00352 3/20 0.56
KDM4E B2RXH2 3/20 0.56
HPGD P15428 1/20 0.56
HSD17B10 Q99714 1/20 0.56
MEN1 O00255 5/20 0.56
KMT2A Q03164 5/20 0.56
HTT P42858 3/20 0.56
LMNA P02545 3/20 0.54
GAA P10253 1/20 0.54
RAB9A P51151 4/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
NPC1 O15118 3/20 0.52
NPSR1 Q6W5P4 2/20 0.52
MAPT P10636 2/20 0.52
L3MBTL1 Q9Y468 2/20 0.52
TDP1 Q9NUW8 1/20 0.52
CYP3A4 P08684 1/20 0.50
ALOX15 P16050 1/20 0.50
TSHR P16473 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8826118 0.87 KDM4E (0.75) DHODHALDH1A1KDM4EHPGDHSD17B10
SCHEMBL2122993 0.85 ALDH1A1 (0.77) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL4611285 0.84 DHODH (0.60) DHODHALDH1A1KDM4EHPGDHSD17B10
SCHEMBL15635912 0.84 KDM4E (0.62) DHODHALDH1A1KDM4EHPGDHSD17B10
SCHEMBL8696115 0.84 DHODH (0.52) DHODHALDH1A1KDM4EHPGDHSD17B10
SCHEMBL1179790 0.83 DHODH (0.55) DHODHALDH1A1KDM4EHPGDHSD17B10
SCHEMBL11492008 0.83 KDM4E (0.54) ALDH1A1KDM4EHPGDHSD17B10HTT
SCHEMBL3569657 0.83 KDM4E (0.54) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL14399048 0.83 DHODH (0.55) DHODHALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9239004 0.83 KDM4E (0.61) DHODHALDH1A1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2804868-B1 PYRAN-SPIROCYCLIC PIPERIDINE AMIDES AS MODULATORS OF ION CHANNELS VERTEX PHARMA (US) 2017-04-12 EP disclosed
US-6914160-B1 Oxytocin inhibitors PFIZER INC (US) 2005-07-05 US disclosed
EP-1537085-A1 OXYTOCIN INHIBITORS Pfizer Limited (GB) 2005-06-08 EP disclosed
WO-2004020414-A1 OXYTOCIN INHIBITORS PFIZER LIMITED (GB) 2004-03-11 WO disclosed
WO-2004020414-A1 OXYTOCIN INHIBITORS PFIZER LIMITED (GB) 2004-03-11 WO disclosed
US-4215123-A Antisecretory 4-oxy-3-carboxy or cyano-1,2-dihydro-2-oxo-1,8-naphthyridine derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1980-07-29 US disclosed